Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 3560
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36357((3R,6R,7S,8E,10S,11S,12E,14E,16S,18R,19R,20R,21S)-...)
Affinity DataEC50:  1nMpH: 7.8 T: 2°CAssay Description:Placental alkaline phosphatase (PLAP) reporter assay controlled by VEGF promoter (VEGF-PLAP)More data for this Ligand-Target Pair
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36358((3R,6R,7S,8E,10S,11S,12E,14E,16R,18R,19R,20R,21S)-...)
Affinity DataEC50:  4.30nMpH: 7.8 T: 2°CAssay Description:Placental alkaline phosphatase (PLAP) reporter assay controlled by VEGF promoter (VEGF-PLAP)More data for this Ligand-Target Pair
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36359((3R,6R,7S,8E,10S,11S,12E,14E,16R,18R,19R,20R,21S)-...)
Affinity DataEC50:  3.60nMpH: 7.8 T: 2°CAssay Description:Placental alkaline phosphatase (PLAP) reporter assay controlled by VEGF promoter (VEGF-PLAP)More data for this Ligand-Target Pair
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36360(CID16202133 | Pladienolide analog 8)
Affinity DataEC50:  4.90nMpH: 7.8 T: 2°CAssay Description:Placental alkaline phosphatase (PLAP) reporter assay controlled by VEGF promoter (VEGF-PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36361(CID16202134 | Pladienolide analog 9)
Affinity DataEC50:  78.4nMpH: 7.8 T: 2°CAssay Description:Placental alkaline phosphatase (PLAP) reporter assay controlled by VEGF promoter (VEGF-PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36362(CID1620213 | Pladienolide analog 10)
Affinity DataEC50:  595nMpH: 7.8 T: 2°CAssay Description:Cell proliferation assay using WiDrMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36357((3R,6R,7S,8E,10S,11S,12E,14E,16S,18R,19R,20R,21S)-...)
Affinity DataEC50:  0.860nMpH: 7.8 T: 2°CAssay Description:Cell proliferation assay using WiDrMore data for this Ligand-Target Pair
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36358((3R,6R,7S,8E,10S,11S,12E,14E,16R,18R,19R,20R,21S)-...)
Affinity DataEC50:  6nMpH: 7.8 T: 2°CAssay Description:Cell proliferation assay using WiDrMore data for this Ligand-Target Pair
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36359((3R,6R,7S,8E,10S,11S,12E,14E,16R,18R,19R,20R,21S)-...)
Affinity DataEC50:  3.20nMpH: 7.8 T: 2°CAssay Description:Cell proliferation assay using WiDrMore data for this Ligand-Target Pair
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36360(CID16202133 | Pladienolide analog 8)
Affinity DataEC50:  6.10nMpH: 7.8 T: 2°CAssay Description:Cell proliferation assay using WiDrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36361(CID16202134 | Pladienolide analog 9)
Affinity DataEC50:  70.2nMpH: 7.8 T: 2°CAssay Description:Cell proliferation assay using WiDrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSplicing factor 3B subunit 3(Homo sapiens (Human))
Eisai

LigandPNGBDBM36361(CID16202134 | Pladienolide analog 9)
Affinity DataEC50:  645nMpH: 7.8 T: 2°CAssay Description:Placental alkaline phosphatase (PLAP) reporter assay controlled by VEGF promoter (VEGF-PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed