Compile Data Set for Download or QSAR
maximum 50k data
Found 96 Enz. Inhib. hit(s) with all data for entry = 50020871
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218471(4-[7,7,10,10-tetramethyl-5-propyl-2-(3-trifluorome...)
Affinity DataIC50:  76nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218455(4-[5-ethyl-7,7,10,10-tetramethyl-2-(3-trifluoromet...)
Affinity DataIC50:  95nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218481(4-[2-(4-fluoro-benzenesulfonylamino)-7,7,10,10-tet...)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218461(4-[2-(butane-1-sulfonylamino)-7,7,10,10-tetramethy...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218455(4-[5-ethyl-7,7,10,10-tetramethyl-2-(3-trifluoromet...)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218468(4-[2-(4-fluoro-benzenesulfonylamino)-5,7,7,10,10-p...)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218471(4-[7,7,10,10-tetramethyl-5-propyl-2-(3-trifluorome...)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218458(4-[2-(butane-1-sulfonylamino)-5-ethyl-7,7,10,10-te...)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218492(4-[5-ethyl-2-(4-fluoro-benzenesulfonylamino)-7,7,1...)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218495(4-[5,7,7,10,10-pentamethyl-2-(propane-1-sulfonylam...)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218458(4-[2-(butane-1-sulfonylamino)-5-ethyl-7,7,10,10-te...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218454(4-[5-ethyl-7,7,10,10-tetramethyl-2-(propane-1-sulf...)
Affinity DataIC50:  340nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218469(4-[2-(butane-1-sulfonylamino)-5,7,7,10,10-pentamet...)
Affinity DataIC50:  370nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218496(4-[5,7,7,10,10-pentamethyl-2-((E)-2-phenyl-ethenes...)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218492(4-[5-ethyl-2-(4-fluoro-benzenesulfonylamino)-7,7,1...)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218499(4-[5,7,7,10,10-pentamethyl-2-(toluene-4-sulfonylam...)
Affinity DataIC50:  430nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218490(4-[2-(4-methoxy-benzenesulfonylamino)-5,7,7,10,10-...)
Affinity DataIC50:  470nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218456(4-[5,7,7,10,10-pentamethyl-2-(3-trifluoromethyl-be...)
Affinity DataIC50:  480nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218466(4-(2-benzenesulfonylamino-5,7,7,10,10-pentamethyl-...)
Affinity DataIC50:  510nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218457(4-[7,7,10,10-tetramethyl-2-(propane-1-sulfonylamin...)
Affinity DataIC50:  550nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218454(4-[5-ethyl-7,7,10,10-tetramethyl-2-(propane-1-sulf...)
Affinity DataIC50:  570nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218472(4-{5-ethyl-2-[2-(4-fluoro-phenyl)-acetylamino]-7,7...)
Affinity DataIC50:  720nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218481(4-[2-(4-fluoro-benzenesulfonylamino)-7,7,10,10-tet...)
Affinity DataIC50:  810nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218476(4-(2-ethanesulfonylamino-5,7,7,10,10-pentamethyl-7...)
Affinity DataIC50:  840nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218457(4-[7,7,10,10-tetramethyl-2-(propane-1-sulfonylamin...)
Affinity DataIC50:  840nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218461(4-[2-(butane-1-sulfonylamino)-7,7,10,10-tetramethy...)
Affinity DataIC50:  850nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218483(4-[5,7,7,10,10-pentamethyl-2-(naphthalene-1-sulfon...)
Affinity DataIC50:  850nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218487(4-{2-[2-(4-fluoro-phenyl)-acetylamino]-5,7,7,10,10...)
Affinity DataIC50:  880nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218464((Z)-4-(5,7,7,10,10-pentamethyl-2-nitro-7,8,9,10-te...)
Affinity DataIC50:  900nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218488(4-(2-benzoylamino-5,7,7,10,10-pentamethyl-7,8,9,10...)
Affinity DataIC50:  900nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218469(4-[2-(butane-1-sulfonylamino)-5,7,7,10,10-pentamet...)
Affinity DataIC50:  910nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218463(4-(5,7,7,10,10-pentamethyl-2-phenylacetylamino-7,8...)
Affinity DataIC50:  970nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218465(4-(5,7,7,10,10-pentamethyl-2-phenylmethanesulfonyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218485(4-[5,7,7,10,10-pentamethyl-2-(4-trifluoromethyl-be...)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218491(4-[2-(3,5-bis-trifluoromethyl-benzenesulfonylamino...)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218472(4-{5-ethyl-2-[2-(4-fluoro-phenyl)-acetylamino]-7,7...)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218464((Z)-4-(5,7,7,10,10-pentamethyl-2-nitro-7,8,9,10-te...)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218482(4-[2-(3-fluoro-benzenesulfonylamino)-5,7,7,10,10-p...)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218487(4-{2-[2-(4-fluoro-phenyl)-acetylamino]-5,7,7,10,10...)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218501(4-[2-(biphenyl-4-sulfonylamino)-5,7,7,10,10-pentam...)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218474(4-[5,7,7,10,10-pentamethyl-2-(2-trifluoromethyl-be...)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218466(4-(2-benzenesulfonylamino-5,7,7,10,10-pentamethyl-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218475(4-[2-(cyclohexanecarbonyl-amino)-5,7,7,10,10-penta...)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218456(4-[5,7,7,10,10-pentamethyl-2-(3-trifluoromethyl-be...)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218470(4-[2-(4-fluoro-benzoylamino)-5,7,7,10,10-pentameth...)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218470(4-[2-(4-fluoro-benzoylamino)-5,7,7,10,10-pentameth...)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218468(4-[2-(4-fluoro-benzenesulfonylamino)-5,7,7,10,10-p...)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218479(4-(2-butyrylamino-5,7,7,10,10-pentamethyl-7,8,9,10...)
Affinity DataIC50:  1.80E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218493(4-(2-isobutyrylamino-5,7,7,10,10-pentamethyl-7,8,9...)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of 9-cis-retinoic acid-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50218488(4-(2-benzoylamino-5,7,7,10,10-pentamethyl-7,8,9,10...)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at human RXRalpha expressed in EK293 cells assessed as inhibition of LG100268-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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