Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50025428
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242808(2-((3,5-bis(trifluoromethyl)benzyl)(4-(3-(trifluor...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242811(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-methyl-3,...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242810(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-(4-(trifl...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242812(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-propyl-3,...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242805(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-(4-(trifl...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242790(2-((3,5-bis(trifluoromethyl)benzyl)(4-(4-(trifluor...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50149275(2-(1-benzyl-5-(4-(trifluoromethoxy)phenyl)-1H-indo...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242809(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-allyl-3-(...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242813(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-allyl-3,5...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242803(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-allyl-4-(...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242774(CHEMBL460054 | N-(3,5-Bis-trifluoromethyl-benzyl)-...)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242802(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-pentyl-4-...)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242791(2-((3,5-bis(trifluoromethyl)benzyl)(4-(3-(trifluor...)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242801(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-propyl-4-...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242773(CHEMBL460053 | N-(4'-Trifluoromethoxy-biphenyl-4-y...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242800(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-methyl-4-...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242789(2-((3,5-bis(trifluoromethyl)benzyl)(4-(3,4-difluor...)
Affinity DataIC50:  2.99E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242804(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-benzyl-4-...)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242807(2-((3,5-bis(trifluoromethyl)benzyl)(4-(N-methyl-4-...)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242787(2-((3,5-bis(trifluoromethyl)benzyl)(4-(4-chlorophe...)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242788(2-((3,5-bis(trifluoromethyl)benzyl)(4-(4-methoxyph...)
Affinity DataIC50: >8.00E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242806(2-((3,5-bis(trifluoromethyl)benzyl)(4-(4-(trifluor...)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242752(CHEMBL459636 | N-Benzyl-N-(4'-trifluoromethoxy-bip...)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50242799(2-((3,5-bis(trifluoromethyl)benzyl)(4-(2-(trifluor...)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of human PAI1 by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed