Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 2564
TargetProtein kinase YpkA(Yersinia pestis)
The Rockefeller University

LigandPNGBDBM22042((3Z)-5-bromo-3-[3-(3-chlorophenyl)-4-oxo-2-thioxo-...)
Affinity DataIC50:  1.81E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22042((3Z)-5-bromo-3-[3-(3-chlorophenyl)-4-oxo-2-thioxo-...)
Affinity DataIC50:  2.45E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase YpkA(Yersinia pestis)
The Rockefeller University

LigandPNGBDBM22045(5-({4-[(4-chlorophenyl)sulfanyl]-3-nitrophenyl}met...)
Affinity DataIC50:  5.87E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase YpkA(Yersinia pestis)
The Rockefeller University

LigandPNGBDBM22044((5Z)-5-{[5-(2-chloro-5-nitrophenyl)furan-2-yl]meth...)
Affinity DataIC50:  9.72E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase YpkA(Yersinia pestis)
The Rockefeller University

LigandPNGBDBM22043(N-(3-nitrophenyl)-9,10-dioxo-9,10-dihydroanthracen...)
Affinity DataIC50:  1.98E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22045(5-({4-[(4-chlorophenyl)sulfanyl]-3-nitrophenyl}met...)
Affinity DataIC50:  5.30E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22044((5Z)-5-{[5-(2-chloro-5-nitrophenyl)furan-2-yl]meth...)
Affinity DataIC50:  5.45E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22043(N-(3-nitrophenyl)-9,10-dioxo-9,10-dihydroanthracen...)
Affinity DataIC50:  1.65E+5nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22042((3Z)-5-bromo-3-[3-(3-chlorophenyl)-4-oxo-2-thioxo-...)
Affinity DataIC50: >2.00E+5nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22045(5-({4-[(4-chlorophenyl)sulfanyl]-3-nitrophenyl}met...)
Affinity DataIC50: >2.00E+5nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22043(N-(3-nitrophenyl)-9,10-dioxo-9,10-dihydroanthracen...)
Affinity DataIC50: >2.00E+5nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22044((5Z)-5-{[5-(2-chloro-5-nitrophenyl)furan-2-yl]meth...)
Affinity DataIC50:  2.05E+5nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed