Compile Data Set for Download or QSAR
maximum 50k data
Found 34 Enz. Inhib. hit(s) with all data for entry = 50021013
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219939(CHEMBL240693 | N-((1r,4r)-4-(2-(4-(2,3-dichlorophe...)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219946(CHEMBL391700 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219943(CHEMBL428910 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219940(CHEMBL240271 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  0.5nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219944(CHEMBL239847 | N-((1r,4r)-4-(2-(4-(4-bromo-2-metho...)
Affinity DataIC50:  0.5nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219947(CHEMBL429093 | N-((1r,4r)-4-(2-(4-(3-cyanophenyl)p...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219945(CHEMBL240273 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219935(CHEMBL392528 | N-[4-(4-{2-[4-(3-cyano-5-trifluorom...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219949(3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)pheno...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219942(CHEMBL240051 | N-((1r,4r)-4-(2-(4-(2,5-dichlorophe...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219948(CHEMBL236407 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219938(CHEMBL391699 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  2.80nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219937(4-chloro-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)ph...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219936(4-bromo-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219934(CHEMBL399833 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  3.80nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219939(CHEMBL240693 | N-((1r,4r)-4-(2-(4-(2,3-dichlorophe...)
Affinity DataIC50:  4nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219941(CHEMBL240909 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219940(CHEMBL240271 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  4.30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219949(3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)pheno...)
Affinity DataIC50:  5.30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219950(3-cyano-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50:  5.80nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219942(CHEMBL240051 | N-((1r,4r)-4-(2-(4-(2,5-dichlorophe...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219937(4-chloro-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)ph...)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219950(3-cyano-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50:  23nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219943(CHEMBL428910 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...)
Affinity DataIC50:  24nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219936(4-bromo-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50:  26nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219944(CHEMBL239847 | N-((1r,4r)-4-(2-(4-(4-bromo-2-metho...)
Affinity DataIC50:  28nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219946(CHEMBL391700 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219945(CHEMBL240273 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219941(CHEMBL240909 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...)
Affinity DataIC50:  39nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219935(CHEMBL392528 | N-[4-(4-{2-[4-(3-cyano-5-trifluorom...)
Affinity DataIC50:  39nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219934(CHEMBL399833 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  41nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219947(CHEMBL429093 | N-((1r,4r)-4-(2-(4-(3-cyanophenyl)p...)
Affinity DataIC50:  57nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219938(CHEMBL391699 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  66nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219948(CHEMBL236407 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...)
Affinity DataIC50:  91nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed