Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50021142
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221444((R)-1-((R)-8-((1H-1,2,4-triazol-1-yl)methyl)-2-(tr...)
Affinity DataIC50:  2nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221449((3R)-1-(8-((1H-imidazol-1-yl)methyl)-2-(trifluorom...)
Affinity DataIC50:  2nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221454((R)-1-((R)-8-(4-(trifluoromethyl)benzyl)-2-(triflu...)
Affinity DataIC50:  4nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221452((R)-1-((R)-8-(4-fluorobenzyl)-2-(trifluoromethyl)-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221442((3R)-1-(8-((1H-pyrazol-1-yl)methyl)-2-(trifluorome...)
Affinity DataIC50:  4nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221453((3R)-1-(8-((1H-1,2,4-triazol-1-yl)methyl)-2-(trifl...)
Affinity DataIC50:  5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221451((R)-3-amino-1-((R)-8-(cyclopropylmethyl)-2-(triflu...)
Affinity DataIC50:  7nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221445((R)-3-amino-1-((R)-8-(cyclopropylfluoromethyl)-2-(...)
Affinity DataIC50:  11nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221445((R)-3-amino-1-((R)-8-(cyclopropylfluoromethyl)-2-(...)
Affinity DataIC50:  11nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221446((R)-3-amino-1-((R)-8-(cyclopropyl(hydroxy)methyl)-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221440((R)-3-amino-1-((R)-8-(cyclopropyl(hydroxy)methyl)-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  18nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221443((2R)-4-[(8R)-8-METHYL-2-(TRIFLUOROMETHYL)-5,6-DIHY...)
Affinity DataIC50:  25nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221447((R)-3-amino-1-(2-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  59nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221448((R)-3-amino-1-(2-phenyl-5,6-dihydro-[1,2,4]triazol...)
Affinity DataIC50:  68nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221441((R)-3-amino-1-(2-cyclopropyl-5,6-dihydro-[1,2,4]tr...)
Affinity DataIC50:  71nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221450((R)-3-amino-1-(5,6-dihydro-[1,2,4]triazolo[1,5-a]p...)
Affinity DataIC50:  100nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221455((R)-3-amino-1-((S)-8-methyl-2-(trifluoromethyl)-5,...)
Affinity DataIC50:  274nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221448((R)-3-amino-1-(2-phenyl-5,6-dihydro-[1,2,4]triazol...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221445((R)-3-amino-1-((R)-8-(cyclopropylfluoromethyl)-2-(...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221445((R)-3-amino-1-((R)-8-(cyclopropylfluoromethyl)-2-(...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221451((R)-3-amino-1-((R)-8-(cyclopropylmethyl)-2-(triflu...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221442((3R)-1-(8-((1H-pyrazol-1-yl)methyl)-2-(trifluorome...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221454((R)-1-((R)-8-(4-(trifluoromethyl)benzyl)-2-(triflu...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221454((R)-1-((R)-8-(4-(trifluoromethyl)benzyl)-2-(triflu...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221440((R)-3-amino-1-((R)-8-(cyclopropyl(hydroxy)methyl)-...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221444((R)-1-((R)-8-((1H-1,2,4-triazol-1-yl)methyl)-2-(tr...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221443((2R)-4-[(8R)-8-METHYL-2-(TRIFLUOROMETHYL)-5,6-DIHY...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221452((R)-1-((R)-8-(4-fluorobenzyl)-2-(trifluoromethyl)-...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221449((3R)-1-(8-((1H-imidazol-1-yl)methyl)-2-(trifluorom...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221454((R)-1-((R)-8-(4-(trifluoromethyl)benzyl)-2-(triflu...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221452((R)-1-((R)-8-(4-fluorobenzyl)-2-(trifluoromethyl)-...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221449((3R)-1-(8-((1H-imidazol-1-yl)methyl)-2-(trifluorom...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221446((R)-3-amino-1-((R)-8-(cyclopropyl(hydroxy)methyl)-...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221448((R)-3-amino-1-(2-phenyl-5,6-dihydro-[1,2,4]triazol...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221453((3R)-1-(8-((1H-1,2,4-triazol-1-yl)methyl)-2-(trifl...)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221451((R)-3-amino-1-((R)-8-(cyclopropylmethyl)-2-(triflu...)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221447((R)-3-amino-1-(2-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221452((R)-1-((R)-8-(4-fluorobenzyl)-2-(trifluoromethyl)-...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221447((R)-3-amino-1-(2-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221445((R)-3-amino-1-((R)-8-(cyclopropylfluoromethyl)-2-(...)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221445((R)-3-amino-1-((R)-8-(cyclopropylfluoromethyl)-2-(...)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221451((R)-3-amino-1-((R)-8-(cyclopropylmethyl)-2-(triflu...)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221455((R)-3-amino-1-((S)-8-methyl-2-(trifluoromethyl)-5,...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of QPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221446((R)-3-amino-1-((R)-8-(cyclopropyl(hydroxy)methyl)-...)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221443((2R)-4-[(8R)-8-METHYL-2-(TRIFLUOROMETHYL)-5,6-DIHY...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221447((R)-3-amino-1-(2-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221449((3R)-1-(8-((1H-imidazol-1-yl)methyl)-2-(trifluorom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221450((R)-3-amino-1-(5,6-dihydro-[1,2,4]triazolo[1,5-a]p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221444((R)-1-((R)-8-((1H-1,2,4-triazol-1-yl)methyl)-2-(tr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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