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Found 18 Enz. Inhib. hit(s) with all data for entry = 50021301
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223074(CHEMBL250466 | N-((6-amino-2-methylpyridin-3-yl)me...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223067(CHEMBL250651 | N-(6-amino-2-methyl-pyridin-3-ylmet...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223066(CHEMBL250650 | N-[2-({[amino(imino)methyl]amino}ox...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223081(CHEMBL250273 | N-[2-(carbamimidamidooxy)ethyl]-2-(...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223071(CHEMBL399868 | N-((6-amino-2-methylpyridin-3-yl)me...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223069(CHEMBL250461 | N-[2-(carbamimidamidooxy)ethyl]-2-(...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223078(CHEMBL250465 | N-((6-amino-2,4-dimethylpyridin-3-y...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223065(CHEMBL250460 | N-[2-(carbamimidamidooxy)ethyl]-2-(...)
Affinity DataKi:  4.70nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223075(CHEMBL250463 | N-[2-({[amino(imino)methyl]amino}ox...)
Affinity DataKi:  8.60nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223076(CHEMBL399662 | N-((6-amino-2-methylpyridin-3-yl)me...)
Affinity DataKi:  10nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223077(CHEMBL250271 | N-[2-({[amino(imino)methyl]amino}ox...)
Affinity DataKi:  34nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223072(CHEMBL401842 | N-[2-(carbamimidamidooxy)ethyl]-2-{...)
Affinity DataKi:  47nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223073(CHEMBL428413 | N-[2-(carbamimidamidooxy)ethyl]-2-[...)
Affinity DataKi:  57nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223068(CHEMBL250274 | N-[2-(carbamimidamidooxy)ethyl]-2-(...)
Affinity DataKi:  58nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223064(CHEMBL250275 | N-[2-(carbamimidamidooxy)ethyl]-2-(...)
Affinity DataKi:  128nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223070(CHEMBL250464 | N-[2-(carbamimidamidooxy)ethyl]-2-[...)
Affinity DataKi:  142nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223079(CHEMBL250649 | N-[2-(carbamimidamidooxy)ethyl]-2-(...)
Affinity DataKi:  169nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50223080(CHEMBL250646 | N-[2-({[amino(imino)methyl]amino}ox...)
Affinity DataKi:  1.28E+3nMAssay Description:Inhibition of human thrombin after 15 mins by standard chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed