Compile Data Set for Download or QSAR
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Found 19 Enz. Inhib. hit(s) with all data for entry = 50021597
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226108(CHEMBL238568 | N-(2-aminophenyl)-4-((4-oxo-4H-chro...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226111(CHEMBL241337 | N-(2-aminophenyl)-4-((2,4-dioxo-1,2...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226109(CHEMBL401449 | N-(2-aminophenyl)-4-((2,4-dioxo-1,2...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226107(CHEMBL400213 | N-(2-aminophenyl)-4-((2-methyl-4-ox...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226117(CHEMBL396444 | N-(2-aminophenyl)-4-((4-oxochroman-...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226115(CHEMBL239625 | N-(2-aminophenyl)-4-((1-oxoisoindol...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226116(4-((1-(4-methoxybenzyl)-2,4-dioxo-1,2-dihydroquina...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226118(CHEMBL241338 | N-(2-aminophenyl)-4-((1-methyl-2,4-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226114(CHEMBL392449 | N-(2-aminophenyl)-4-((4-oxoquinazol...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226120(CHEMBL398394 | N-(2-aminophenyl)-4-((1-oxo-2,3-dih...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226112(CHEMBL400419 | N-(2-aminophenyl)-4-((2,4-dioxo-2H-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226124(CHEMBL240915 | N-(2-aminophenyl)-4-((4-oxobenzo[d]...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226123(CHEMBL241549 | N-(2-aminophenyl)-4-((1-ethyl-2,4-d...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226106(CHEMBL241757 | N-(2-aminophenyl)-4-((4-oxothieno[3...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226110(CHEMBL241129 | N-(2-aminophenyl)-4-((1,3-dioxoisoi...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226119(CHEMBL241759 | N-(2-aminophenyl)-4-((1-ethyl-2,4-d...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226121(CHEMBL401448 | N-(2-aminophenyl)-4-((1-(2-(dimethy...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226122(CHEMBL241550 | N-(2-aminophenyl)-4-((1-(2-morpholi...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50226113(CHEMBL238569 | N-(2-aminophenyl)-4-(chroman-3-ylme...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant HDAC1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed