Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 50025605
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  130nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247392(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  150nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  150nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  150nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  150nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  160nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247393(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  170nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247396(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  260nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247417(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  280nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247394(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  300nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  450nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247431(CHEMBL461739 | N-Benzyl-8-isopopyl-9-oxo-8,9-dihyd...)
Affinity DataIC50:  520nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186073(CHEMBL210229 | N-(2-(dimethylamino)ethyl)-8-isopro...)
Affinity DataIC50:  560nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247391(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  640nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186084(CHEMBL210474 | N-(2-(dimethylamino)ethyl)-8-ethyl-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247393(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247392(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247394(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247372(8-Ethyl-9-oxo-8,9-dihydro-6-thiazolo[5,4-f]quinazo...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247419(CHEMBL454130 | N-Benzyl-8-ethyl-9-oxo-8,9-dihydrot...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247417(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186073(CHEMBL210229 | N-(2-(dimethylamino)ethyl)-8-isopro...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247394(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247391(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247396(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186082(8-ethyl-N-isopropyl-9-oxo-8,9-dihydrothiazolo[5,4-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247431(CHEMBL461739 | N-Benzyl-8-isopopyl-9-oxo-8,9-dihyd...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247431(CHEMBL461739 | N-Benzyl-8-isopopyl-9-oxo-8,9-dihyd...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186072(CHEMBL378190 | N,8-diisopropyl-9-oxo-8,9-dihydroth...)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186073(CHEMBL210229 | N-(2-(dimethylamino)ethyl)-8-isopro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247419(CHEMBL454130 | N-Benzyl-8-ethyl-9-oxo-8,9-dihydrot...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186073(CHEMBL210229 | N-(2-(dimethylamino)ethyl)-8-isopro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186084(CHEMBL210474 | N-(2-(dimethylamino)ethyl)-8-ethyl-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247372(8-Ethyl-9-oxo-8,9-dihydro-6-thiazolo[5,4-f]quinazo...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247372(8-Ethyl-9-oxo-8,9-dihydro-6-thiazolo[5,4-f]quinazo...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247393(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247419(CHEMBL454130 | N-Benzyl-8-ethyl-9-oxo-8,9-dihydrot...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186072(CHEMBL378190 | N,8-diisopropyl-9-oxo-8,9-dihydroth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247431(CHEMBL461739 | N-Benzyl-8-isopopyl-9-oxo-8,9-dihyd...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186082(8-ethyl-N-isopropyl-9-oxo-8,9-dihydrothiazolo[5,4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed