Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 2718
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23763(3-({4-[(4-icosylpiperazin-1-yl)carbonyl]phenyl}met...)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23764(3-({4-[(4-docosylpiperazin-1-yl)carbonyl]phenyl}me...)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  470nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23762(3-({4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50:  800nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23759(3-{4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50:  1.10E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23756(3-({4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50:  2.20E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23767(3-{[4-(4-octadecylpiperazin-1-yl)phenyl]methyl}-4,...)
Affinity DataIC50:  2.71E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23766(3-{[4-(4-hexadecylpiperazin-1-yl)phenyl]methyl}-4,...)
Affinity DataIC50:  3.50E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23770(3-{[4-(tetradecyloxy)phenyl]methyl}-4,5-dihydro-1,...)
Affinity DataIC50:  4.00E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23761(3-({4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50:  4.00E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23765(3-{[4-(4-tetradecylpiperazin-1-yl)phenyl]methyl}-4...)
Affinity DataIC50:  4.50E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23753(3-{4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50:  5.08E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23769(3-(3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phen...)
Affinity DataIC50:  5.30E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  8.00E+3nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23760(3-({4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl...)
Affinity DataIC50:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23754(3-({4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}m...)
Affinity DataIC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23755(3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50:  1.00E+4nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23768(3-(2-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phen...)
Affinity DataIC50:  1.87E+4nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23766(3-{[4-(4-hexadecylpiperazin-1-yl)phenyl]methyl}-4,...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23767(3-{[4-(4-octadecylpiperazin-1-yl)phenyl]methyl}-4,...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23768(3-(2-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phen...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23769(3-(3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phen...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23770(3-{[4-(tetradecyloxy)phenyl]methyl}-4,5-dihydro-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23765(3-{[4-(4-tetradecylpiperazin-1-yl)phenyl]methyl}-4...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23764(3-({4-[(4-docosylpiperazin-1-yl)carbonyl]phenyl}me...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23763(3-({4-[(4-icosylpiperazin-1-yl)carbonyl]phenyl}met...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23762(3-({4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23761(3-({4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23760(3-({4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23759(3-{4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23758(3-{4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23757(3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23756(3-({4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23755(3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23754(3-({4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}m...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23753(3-{4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23752(3-{4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23750(3-{4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}-4...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23758(3-{4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23757(3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23750(3-{4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}-4...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23752(3-{4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed