Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50025614
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264513(4-Bromo-6-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-e...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264478(4-Chloro-6-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-...)
Affinity DataKi:  5.49nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264541(4-Bromo-6-(2-{4-[3-(trifluoromethyl)phenyl]piperaz...)
Affinity DataKi:  5.77nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264544(6-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-1H-...)
Affinity DataKi:  13.1nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264509(4-Chloro-6-{2-[4-(2-chlorophenyl)piperazin-1-yl]et...)
Affinity DataKi:  19.1nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264542(4-Bromo-6-{2-[4-(2-pyrimidinyl)piperazin-1-yl]ethy...)
Affinity DataKi:  26.7nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264568(6-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)-1H-b...)
Affinity DataKi:  59.7nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264512(4-Bromo-6-[2-(4-phenylpiperazin-1-yl)ethyl]-1H-ben...)
Affinity DataKi:  61.9nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264477(4-Chloro-6-[2-(4-phenylpiperazin-1-yl)ethyl]-1H-be...)
Affinity DataKi:  84.7nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264540(4-Bromo-6-{2-[4-(2-chlorophenyl)piperazin-1-yl]eth...)
Affinity DataKi:  84.7nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264543(6-(2-(4-phenylpiperazin-1-yl)ethyl)-1H-benzo[d]imi...)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264510(4-Chloro-6-(2-{4-[3-(trifluoromethyl)phenyl]pipera...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264569(6-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)...)
Affinity DataKi:  273nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264511(4-Chloro-6-{2-[4-(2-pyrimidinyl)piperazin-1-yl]eth...)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264510(4-Chloro-6-(2-{4-[3-(trifluoromethyl)phenyl]pipera...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264511(4-Chloro-6-{2-[4-(2-pyrimidinyl)piperazin-1-yl]eth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264512(4-Bromo-6-[2-(4-phenylpiperazin-1-yl)ethyl]-1H-ben...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264513(4-Bromo-6-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-e...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264540(4-Bromo-6-{2-[4-(2-chlorophenyl)piperazin-1-yl]eth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264541(4-Bromo-6-(2-{4-[3-(trifluoromethyl)phenyl]piperaz...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264542(4-Bromo-6-{2-[4-(2-pyrimidinyl)piperazin-1-yl]ethy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264543(6-(2-(4-phenylpiperazin-1-yl)ethyl)-1H-benzo[d]imi...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264569(6-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264477(4-Chloro-6-[2-(4-phenylpiperazin-1-yl)ethyl]-1H-be...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264570(6-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)-1H-b...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264509(4-Chloro-6-{2-[4-(2-chlorophenyl)piperazin-1-yl]et...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50264478(4-Chloro-6-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed