Compile Data Set for Download or QSAR
maximum 50k data
Found 97 Enz. Inhib. hit(s) with all data for entry = 50037999
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228427((R)-N-[(S)-1-(4-guanidino-benzylcarbamoyl)-ethyl]-...)
Affinity DataKi:  16nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228427((R)-N-[(S)-1-(4-guanidino-benzylcarbamoyl)-ethyl]-...)
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of human recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228427((R)-N-[(S)-1-(4-guanidino-benzylcarbamoyl)-ethyl]-...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228418(CHEMBL393591 | methyl 1-(diphenoxyphosphoryl)-2-(4...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228425(CHEMBL239118 | di-(4-acetamidophenyl) 1-(methylsul...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228420(CHEMBL391968 | di-(4-acetamidophenyl) 1-(benzyloxy...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228421(CHEMBL238493 | diphenyl 1-(methylsulfonylamino)-2-...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228410(CHEMBL239535 | diphenyl 1-(benzyloxycarbonylamino)...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228414(CHEMBL239747 | diphenyl 1-acetamido-2-(4-guanidino...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228417(CHEMBL238491 | diphenyl 1-(o-toluenesulfonylamino)...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  8nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228423(CHEMBL239536 | ethyl 1-(diphenoxyphosphoryl)-2-(4-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Rattus norvegicus)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228418(CHEMBL393591 | methyl 1-(diphenoxyphosphoryl)-2-(4...)
Affinity DataIC50:  19.5nMAssay Description:Inhibition of rat uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Rattus norvegicus)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  24.5nMAssay Description:Inhibition of rat uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228426(CHEMBL391344 | diphenyl 1-(naphthalenesulfonylamin...)
Affinity DataIC50:  26.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228418(CHEMBL393591 | methyl 1-(diphenoxyphosphoryl)-2-(4...)
Affinity DataIC50:  32nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228413(CHEMBL238708 | [1-Benzyloxycarbonylamino-2-(4-carb...)
Affinity DataIC50:  67nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228424(CHEMBL393592 | diphenyl 1-(benzoylamino)-2-(4-guan...)
Affinity DataIC50:  114nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228411(CHEMBL391916 | diphenyl 1-(2,3,6-tri-isopropylbenz...)
Affinity DataIC50:  260nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228415(CHEMBL238707 | [Benzyloxycarbonylamino-(4-carbamim...)
Affinity DataIC50:  288nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228420(CHEMBL391968 | di-(4-acetamidophenyl) 1-(benzyloxy...)
Affinity DataIC50:  390nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  770nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228416(CHEMBL239331 | diphenyl N-(benzyloxycarbonylamino)...)
Affinity DataIC50:  780nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228416(CHEMBL239331 | diphenyl N-(benzyloxycarbonylamino)...)
Affinity DataIC50:  840nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228420(CHEMBL391968 | di-(4-acetamidophenyl) 1-(benzyloxy...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228419(CHEMBL238913 | diphenyl 1-(N-benzyloxycarbonylamin...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228413(CHEMBL238708 | [1-Benzyloxycarbonylamino-2-(4-carb...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228426(CHEMBL391344 | diphenyl 1-(naphthalenesulfonylamin...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228428(CHEMBL238706 | diphenyl 1-amino-2-(4-guanidinophen...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228425(CHEMBL239118 | di-(4-acetamidophenyl) 1-(methylsul...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of rat plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228425(CHEMBL239118 | di-(4-acetamidophenyl) 1-(methylsul...)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228410(CHEMBL239535 | diphenyl 1-(benzyloxycarbonylamino)...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228410(CHEMBL239535 | diphenyl 1-(benzyloxycarbonylamino)...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228415(CHEMBL238707 | [Benzyloxycarbonylamino-(4-carbamim...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228425(CHEMBL239118 | di-(4-acetamidophenyl) 1-(methylsul...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228423(CHEMBL239536 | ethyl 1-(diphenoxyphosphoryl)-2-(4-...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228413(CHEMBL238708 | [1-Benzyloxycarbonylamino-2-(4-carb...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Mus musculus)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of mouse thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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