Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50038194
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373019(CHEMBL270836)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373027(CHEMBL401712)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373021(CHEMBL401616)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373022(CHEMBL256013)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373023(CHEMBL404439)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373020(CHEMBL270835)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373021(CHEMBL401616)
Affinity DataEC50:  1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARdelta expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373021(CHEMBL401616)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at mouse PPARalpha by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373024(CHEMBL447533)
Affinity DataEC50:  100nMAssay Description:Agonist activity at mouse PPARalpha by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373024(CHEMBL447533)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at mouse PPARgamma by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373025(CHEMBL401811)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373025(CHEMBL401811)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373025(CHEMBL401811)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARdelta expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373026(CHEMBL271873)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373024(CHEMBL447533)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373027(CHEMBL401712)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373022(CHEMBL256013)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373023(CHEMBL404439)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373026(CHEMBL271873)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373024(CHEMBL447533)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373020(CHEMBL270835)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARalpha expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed