Compile Data Set for Download or QSAR
maximum 50k data
Found 125 Enz. Inhib. hit(s) with all data for entry = 50041588
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  14.1nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  14.1nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  17.8nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  17.8nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  18.2nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  18.2nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412180(CHEMBL541671)
Affinity DataKi:  19.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412180(CHEMBL541671)
Affinity DataKi:  19.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412174(CHEMBL557808)
Affinity DataKi:  21.9nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  25.1nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  25.1nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  30.2nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  30.2nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  33.1nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  33.1nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412174(CHEMBL557808)
Affinity DataKi:  34.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412173(CHEMBL496915)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412173(CHEMBL496915)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412173(CHEMBL496915)
Affinity DataKi:  38.0nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412173(CHEMBL496915)
Affinity DataKi:  38.0nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  41.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412180(CHEMBL541671)
Affinity DataKi:  41.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412180(CHEMBL541671)
Affinity DataKi:  41.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  41.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  42.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  42.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  42.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  42.7nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  51.3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412184(CHEMBL539373)
Affinity DataKi:  51.3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412180(CHEMBL541671)
Affinity DataKi:  57.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412180(CHEMBL541671)
Affinity DataKi:  57.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  58.9nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  58.9nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  64.6nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  64.6nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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