TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataKi: <0.5nMAssay Description:Binding affinity to BH3 binding groove of BclXLMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to DPP4More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase beta(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to DPP4More data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase catalytic subunit 1(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
TargetQueuine tRNA-ribosyltransferase catalytic subunit 1(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataKi: 7.30E+3nMAssay Description:Binding affinity nNOSMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity to DPP4More data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of aurora kinase AMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of aurora kinase AMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Binding affinity to BH3 binding groove of BclXLMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of aurora kinase AMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Binding affinity to DPP4More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of protein kinase BMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of protein kinase BMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+5nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+6nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Activity against estrogen receptor alphaMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+5nMAssay Description:Binding affinity to HSP90More data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity to HSP90More data for this Ligand-Target Pair
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to HSP90More data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Inhibition of bovine carbonic anhydrase2More data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Inhibition of bovine carbonic anhydrase2More data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataKd: 2.00E+6nMAssay Description:Binding affinity to BH3 binding groove of BclXLMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Activity against estrogen receptor alphaMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataKd: 4.00E+5nMAssay Description:Binding affinity to BH3 binding groove of BclXLMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Activity against estrogen receptor alphaMore data for this Ligand-Target Pair