Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50026315
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244240((20S)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.0260nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50412386(CHEMBL2021486)
Affinity DataEC50:  0.0300nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50005618(CHEMBL2021484)
Affinity DataEC50:  0.00210nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244241((20R)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.200nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244165((1R,2S,3R,5Z,7E)-17-{(1R)-1-[(2-ethyl-2-hydroxybut...)
Affinity DataEC50:  0.0240nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244269((20R)-1-alpha-2-alpha-25-Trihydroxy-2-beta-methyl-...)
Affinity DataEC50:  0.120nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50412386(CHEMBL2021486)
Affinity DataEC50:  0.0580nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244241((20R)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.0290nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244165((1R,2S,3R,5Z,7E)-17-{(1R)-1-[(2-ethyl-2-hydroxybut...)
Affinity DataEC50:  0.115nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244268((20S)-1-alpha-2-alpha-25-Trihydroxy-2beta-methyl-1...)
Affinity DataEC50:  1.90nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244269((20R)-1-alpha-2-alpha-25-Trihydroxy-2-beta-methyl-...)
Affinity DataEC50:  4.5nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244164((20S)-1-alpha-25-Dihydroxy-2-alpha-(2-hydroxyethox...)
Affinity DataEC50:  0.0270nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244268((20S)-1-alpha-2-alpha-25-Trihydroxy-2beta-methyl-1...)
Affinity DataEC50:  0.0170nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50244240((20S)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.0850nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50412385(CHEMBL2021488)
Affinity DataEC50:  0.0900nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50412385(CHEMBL2021488)
Affinity DataEC50:  0.0900nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed