Compile Data Set for Download or QSAR
maximum 50k data
Found 97 Enz. Inhib. hit(s) with all data for entry = 50026355
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50:  1nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243221(2-(4-((4-(5-(6-methoxypyridin-3-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243215(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243219(2-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-triazol...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243220(3-phenyl-2-(4-((4-(5-(pyrazin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243286(CHEMBL499554 | N,N-dimethyl-2-(4-(2-phenyl-3-(4-((...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243285(2-(4-(2-phenyl-3-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243215(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243221(2-(4-((4-(5-(6-methoxypyridin-3-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243284(6-(4-methylpiperazin-1-yl)-2-phenyl-3-(4-((4-(5-(p...)
Affinity DataIC50:  18nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243275(5-(5-(1-((4-(2-(4-methylpiperazin-1-yl)-6-phenylpy...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243220(3-phenyl-2-(4-((4-(5-(pyrazin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  21nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243272(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243215(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  26nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243219(2-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-triazol...)
Affinity DataIC50:  26nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243219(2-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-triazol...)
Affinity DataIC50:  33nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243283(CHEMBL455071 | Dimethyl-(2-{4-[7-(4-{4-[5-(1-oxy-p...)
Affinity DataIC50:  33nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243274(CHEMBL505848 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243273(2-(4-(6-phenyl-7-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2...)
Affinity DataIC50:  37nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243277(5-(5-(1-((4-(2-(4-(2-(dimethylamino)ethyl)piperazi...)
Affinity DataIC50:  37nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243276(2-(4-(7-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-t...)
Affinity DataIC50:  38nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  39nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243272(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243221(2-(4-((4-(5-(6-methoxypyridin-3-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243286(CHEMBL499554 | N,N-dimethyl-2-(4-(2-phenyl-3-(4-((...)
Affinity DataIC50:  43nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50:  44nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243220(3-phenyl-2-(4-((4-(5-(pyrazin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  44nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243285(2-(4-(2-phenyl-3-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  48nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243287(6-(4-methylpiperazin-1-yl)-2-phenyl-3-(4-((4-(5-(p...)
Affinity DataIC50:  52nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50:  62nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243282(2-{4-[7-(4-{4-[5-(1-Oxy-pyridin-4-yl)-4H-[1,2,4]tr...)
Affinity DataIC50:  67nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243283(CHEMBL455071 | Dimethyl-(2-{4-[7-(4-{4-[5-(1-oxy-p...)
Affinity DataIC50:  68nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50:  69nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243280(5-(5-(1-((4-(2-(4-(2-(dimethylamino)ethyl)piperazi...)
Affinity DataIC50:  69nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243290(5-(5-(1-((4-(6-(4-methylpiperazin-1-yl)-2-phenylpy...)
Affinity DataIC50:  70nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243278(5-(5-(1-((4-(2-(4-methylpiperazin-1-yl)-6-phenylpy...)
Affinity DataIC50:  71nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243288(2-(4-(2-phenyl-3-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2...)
Affinity DataIC50:  72nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243273(2-(4-(6-phenyl-7-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243275(5-(5-(1-((4-(2-(4-methylpiperazin-1-yl)-6-phenylpy...)
Affinity DataIC50:  84nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243281(2-(4-Methyl-piperazin-1-yl)-7-(4-{4-[5-(1-oxy-pyri...)
Affinity DataIC50:  88nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243284(6-(4-methylpiperazin-1-yl)-2-phenyl-3-(4-((4-(5-(p...)
Affinity DataIC50:  92nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243280(5-(5-(1-((4-(2-(4-(2-(dimethylamino)ethyl)piperazi...)
Affinity DataIC50:  98nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243289(CHEMBL506827 | N,N-dimethyl-2-(4-(2-phenyl-3-(4-((...)
Affinity DataIC50:  104nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243291(2-(4-(3-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-t...)
Affinity DataIC50:  115nMAssay Description:Inhibition of Akt1 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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