Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50026375
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243356(CHEMBL508659 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  4.30nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243233(CHEMBL487276 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  9nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243449(CHEMBL456875 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  21nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243403(CHEMBL510547 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  26nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243307(CHEMBL453581 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  36nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243309(CHEMBL451773 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  38nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243405(CHEMBL452794 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  55nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243355(CHEMBL452531 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  146nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243448(CHEMBL517102 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  235nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243234(CHEMBL487259 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  311nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243235(CHEMBL488045 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  390nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243404(CHEMBL452027 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  401nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243357(CHEMBL453314 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  542nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243451(CHEMBL460684 | N-(3,5-dimethoxybenzyl)-5-phenyltet...)
Affinity DataIC50:  780nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243308(CHEMBL454087 | N-[3,5-Bis(trifluoromethyl)benzyl]-...)
Affinity DataIC50:  1.23E+3nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50243450(CHEMBL460683 | N-(2-Methoxybenzyl)-5-phenyltetrazo...)
Affinity DataIC50:  2.75E+3nMAssay Description:Displacement of [125I]BH-SP to human recombinant NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed