TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 376nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR7Checked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 8.18E+3nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR5Checked by AuthorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.23E+4nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR6Checked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.50E+4nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.72E+4nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR5Checked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 6.20E+4nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 9.50E+4nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR6Checked by AuthorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR7Checked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.40E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.80E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 2.90E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 2.90E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 4.10E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 4.50E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 6.80E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: 3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT2 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT2 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT3 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT2 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT2 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT2 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT2 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT2 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT2 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT3 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT3 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair