Compile Data Set for Download or QSAR
maximum 50k data
Found 71 Enz. Inhib. hit(s) with all data for entry = 50026669
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262214((2-((1H-indazol-6-yl)methylamino)phenyl)(5-methyl-...)
Affinity DataIC50:  52nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  74nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262274((2-((1H-indazol-6-yl)methylamino)phenyl)(6-methyl-...)
Affinity DataIC50:  76nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  100nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  120nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50:  130nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262057((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50:  140nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262105((5-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  160nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262057((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262106((1,5-dimethyl-1H-indol-3-yl)(2-(quinolin-6-ylmethy...)
Affinity DataIC50:  180nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50:  230nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262056((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50:  240nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262274((2-((1H-indazol-6-yl)methylamino)phenyl)(6-methyl-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262054((2-((1H-indazol-6-yl)methylamino)phenyl)(1-methyl-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262278((2-((1H-indazol-6-yl)methylamino)phenyl)(6-fluoro-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262277((2-((1H-indazol-6-yl)methylamino)phenyl)(5-fluoro-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  270nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50:  300nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262054((2-((1H-indazol-6-yl)methylamino)phenyl)(1-methyl-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262007((2-((1H-benzo[d]imidazol-5-yl)methylamino)phenyl)(...)
Affinity DataIC50:  310nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262275((2-((1H-indazol-6-yl)methylamino)phenyl)(7-methyl-...)
Affinity DataIC50:  355nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262157((5-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50:  450nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  460nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262106((1,5-dimethyl-1H-indol-3-yl)(2-(quinolin-6-ylmethy...)
Affinity DataIC50:  540nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262213((5-chloro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  560nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262009((2-((1H-indazol-6-yl)methylamino)phenyl)(1-(2-meth...)
Affinity DataIC50:  560nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262056((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50:  610nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262158((6-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50:  660nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262108((7-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  700nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  730nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262107((6-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  730nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  800nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262212((6-fluoro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  810nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262331((2-((1H-indazol-6-yl)methylamino)phenyl)(5-chloro-...)
Affinity DataIC50:  830nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261904((1H-indazol-3-yl)(2-(pyridin-4-ylmethylamino)pheny...)
Affinity DataIC50:  870nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262214((2-((1H-indazol-6-yl)methylamino)phenyl)(5-methyl-...)
Affinity DataIC50:  870nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262107((6-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  940nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262275((2-((1H-indazol-6-yl)methylamino)phenyl)(7-methyl-...)
Affinity DataIC50:  950nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262058((1H-indol-3-yl)(2-(quinolin-6-ylmethylamino)phenyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262211((5-fluoro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262331((2-((1H-indazol-6-yl)methylamino)phenyl)(5-chloro-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262278((2-((1H-indazol-6-yl)methylamino)phenyl)(6-fluoro-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261904((1H-indazol-3-yl)(2-(pyridin-4-ylmethylamino)pheny...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262277((2-((1H-indazol-6-yl)methylamino)phenyl)(5-fluoro-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262009((2-((1H-indazol-6-yl)methylamino)phenyl)(1-(2-meth...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262212((6-fluoro-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262105((5-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262157((5-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261904((1H-indazol-3-yl)(2-(pyridin-4-ylmethylamino)pheny...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262158((6-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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