Compile Data Set for Download or QSAR
maximum 50k data
Found 131 Enz. Inhib. hit(s) with all data for entry = 50026689
LigandPNGBDBM50262173(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  16nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262174(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  17nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261783(5,5-dimethyl-2-(6-(pyridin-3-yl)-2,3-dihydrobenzo[...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261838(6,6-dimethyl-2-(6-(6-methylpyridin-3-yl)-2,3-dihyd...)
Affinity DataIC50:  21nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262173(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  22nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261839(5,5-dimethyl-2-(6-(6-methylpyridin-3-yl)-2,3-dihyd...)
Affinity DataIC50:  26nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261838(6,6-dimethyl-2-(6-(6-methylpyridin-3-yl)-2,3-dihyd...)
Affinity DataIC50:  28nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2,3-d...)
Affinity DataIC50:  32nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262225(5,5-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2,3-d...)
Affinity DataIC50:  49nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262169(6,6-dimethyl-2-(6-phenyl-2,3-dihydrobenzo[b][1,4]o...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262176(6,6-dimethyl-2-(6-(2-methyl-1H-imidazol-4-yl)-2,3-...)
Affinity DataIC50:  51nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262225(5,5-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2,3-d...)
Affinity DataIC50:  52nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261839(5,5-dimethyl-2-(6-(6-methylpyridin-3-yl)-2,3-dihyd...)
Affinity DataIC50:  73nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261782(5,5-dimethyl-2-(6-(pyridin-2-yl)-2,3-dihydrobenzo[...)
Affinity DataIC50:  74nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262174(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  77nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2,3-d...)
Affinity DataIC50:  78nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261786(5,5-dimethyl-2-(6-phenyl-2,3-dihydrobenzo[b][1,4]o...)
Affinity DataIC50:  80nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262169(6,6-dimethyl-2-(6-phenyl-2,3-dihydrobenzo[b][1,4]o...)
Affinity DataIC50:  80nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262172(2-(6-(1H-imidazol-5-yl)-2,3-dihydrobenzo[b][1,4]ox...)
Affinity DataIC50:  81nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262173(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  89nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262175(2-(6-(1H-pyrazol-5-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  90nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261837(5,5-dimethyl-2-(6-(pyridin-4-yl)-2,3-dihydrobenzo[...)
Affinity DataIC50:  94nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261841(6,6-dimethyl-2-(6-(6-methylpyridazin-3-yl)-2,3-dih...)
Affinity DataIC50:  107nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262176(6,6-dimethyl-2-(6-(2-methyl-1H-imidazol-4-yl)-2,3-...)
Affinity DataIC50:  107nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261783(5,5-dimethyl-2-(6-(pyridin-3-yl)-2,3-dihydrobenzo[...)
Affinity DataIC50:  113nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261838(6,6-dimethyl-2-(6-(6-methylpyridin-3-yl)-2,3-dihyd...)
Affinity DataIC50:  116nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261840(6,6-dimethyl-2-(6-(pyrimidin-2-yl)-2,3-dihydrobenz...)
Affinity DataIC50:  123nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261841(6,6-dimethyl-2-(6-(6-methylpyridazin-3-yl)-2,3-dih...)
Affinity DataIC50:  139nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262175(2-(6-(1H-pyrazol-5-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  145nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261784(2-(6-bromo-2,3-dihydrobenzo[b][1,4]oxazin-4-yl)-6,...)
Affinity DataIC50:  153nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262170(2-(6-cyclopropyl-2,3-dihydrobenzo[b][1,4]oxazin-4-...)
Affinity DataIC50:  155nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262173(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  156nMAssay Description:Inhibition of PI3K beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261837(5,5-dimethyl-2-(6-(pyridin-4-yl)-2,3-dihydrobenzo[...)
Affinity DataIC50:  159nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262172(2-(6-(1H-imidazol-5-yl)-2,3-dihydrobenzo[b][1,4]ox...)
Affinity DataIC50:  163nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261839(5,5-dimethyl-2-(6-(6-methylpyridin-3-yl)-2,3-dihyd...)
Affinity DataIC50:  164nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261783(5,5-dimethyl-2-(6-(pyridin-3-yl)-2,3-dihydrobenzo[...)
Affinity DataIC50:  172nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262174(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  188nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261840(6,6-dimethyl-2-(6-(pyrimidin-2-yl)-2,3-dihydrobenz...)
Affinity DataIC50:  189nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262170(2-(6-cyclopropyl-2,3-dihydrobenzo[b][1,4]oxazin-4-...)
Affinity DataIC50:  210nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262226(2-(7-methoxy-2,3-dihydrobenzo[b][1,4]oxazin-4-yl)-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261785(2-(6-bromo-2,3-dihydrobenzo[b][1,4]oxazin-4-yl)-5,...)
Affinity DataIC50:  249nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261782(5,5-dimethyl-2-(6-(pyridin-2-yl)-2,3-dihydrobenzo[...)
Affinity DataIC50:  258nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262223(6,6-dimethyl-2-(6-(1-methyl-1H-imidazol-2-yl)-2,3-...)
Affinity DataIC50:  285nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262225(5,5-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2,3-d...)
Affinity DataIC50:  294nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2,3-d...)
Affinity DataIC50:  295nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262174(2-(6-(1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxa...)
Affinity DataIC50:  298nMAssay Description:Inhibition of PI3K beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261839(5,5-dimethyl-2-(6-(6-methylpyridin-3-yl)-2,3-dihyd...)
Affinity DataIC50:  308nMAssay Description:Inhibition of PI3K beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262167(2-(6-acetyl-2,3-dihydrobenzo[b][1,4]oxazin-4-yl)-6...)
Affinity DataIC50:  318nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261784(2-(6-bromo-2,3-dihydrobenzo[b][1,4]oxazin-4-yl)-6,...)
Affinity DataIC50:  321nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262176(6,6-dimethyl-2-(6-(2-methyl-1H-imidazol-4-yl)-2,3-...)
Affinity DataIC50:  325nMAssay Description:Inhibition of PI3K beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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