Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50027376
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50171897((2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | ...)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275748((+/-)-2-(4-chlorophenoxy)-3-(2-chlorophenyl)propan...)
Affinity DataEC50:  2.18E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275748((+/-)-2-(4-chlorophenoxy)-3-(2-chlorophenyl)propan...)
Affinity DataEC50:  2.23E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275749((+/-)-3-(2-bromophenyl)-2-(4-chlorophenoxy)propano...)
Affinity DataEC50:  2.48E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275750((+/-)-2-(4-chlorophenoxy)-3-o-tolylpropanoic acid ...)
Affinity DataEC50:  8.54E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275751(2-(4-chlorophenoxy)-3-(2-propylphenyl)propanoic ac...)
Affinity DataEC50:  3.68E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275804((+/-)-2-(4-chlorophenoxy)-3-(2-(trifluoromethyl)ph...)
Affinity DataEC50:  4.03E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275862((+/-)-4,4'-(2-(prop-1-en-2-yl)propane-1,3-diyl)bis...)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275863((+/-)-3-(4-bromophenyl)-2-(4-chlorophenoxy)propano...)
Affinity DataEC50:  2.07E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275864((+/-)-2-(4-chlorophenoxy)-3-p-tolylpropanoic acid ...)
Affinity DataEC50:  4.36E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275865(2-(4-chlorophenoxy)-3-(4-propylphenyl)propanoic ac...)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275867((+/-)-2-(4-chlorophenoxy)-3-(3-phenoxyphenyl)propa...)
Affinity DataEC50:  3.06E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275920((+/-)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propa...)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275921((R)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275922((S)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  870nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275923((S)-3-(biphenyl-4-yl)-2-(4-chlorophenoxy)propanoic...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275924((S)-2-(4-chlorophenoxy)-3-(4-(thiophen-2-yl)phenyl...)
Affinity DataEC50:  590nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275968((S)-2-(4-chlorophenoxy)-3-(4-(trifluoromethyl)phen...)
Affinity DataEC50:  3.65E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275749((+/-)-3-(2-bromophenyl)-2-(4-chlorophenoxy)propano...)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275750((+/-)-2-(4-chlorophenoxy)-3-o-tolylpropanoic acid ...)
Affinity DataEC50:  9.25E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275751(2-(4-chlorophenoxy)-3-(2-propylphenyl)propanoic ac...)
Affinity DataEC50:  1.43E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275804((+/-)-2-(4-chlorophenoxy)-3-(2-(trifluoromethyl)ph...)
Affinity DataEC50:  2.49E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275805((+/-)-2-(4-chlorophenoxy)-3-(2-phenoxyphenyl)propa...)
Affinity DataEC50:  1.14E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275862((+/-)-4,4'-(2-(prop-1-en-2-yl)propane-1,3-diyl)bis...)
Affinity DataEC50:  2.23E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275863((+/-)-3-(4-bromophenyl)-2-(4-chlorophenoxy)propano...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275864((+/-)-2-(4-chlorophenoxy)-3-p-tolylpropanoic acid ...)
Affinity DataEC50:  2.81E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275865(2-(4-chlorophenoxy)-3-(4-propylphenyl)propanoic ac...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275866(2-(4-chlorophenoxy)-3-(4-hexylphenyl)propanoic aci...)
Affinity DataEC50:  450nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275867((+/-)-2-(4-chlorophenoxy)-3-(3-phenoxyphenyl)propa...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275920((+/-)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propa...)
Affinity DataEC50:  64nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275921((R)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275922((S)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275923((S)-3-(biphenyl-4-yl)-2-(4-chlorophenoxy)propanoic...)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275924((S)-2-(4-chlorophenoxy)-3-(4-(thiophen-2-yl)phenyl...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275968((S)-2-(4-chlorophenoxy)-3-(4-(trifluoromethyl)phen...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50171897((2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | ...)
Affinity DataEC50:  1.45E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275697((+/-)-2-(2,4-dichlorophenoxy)-3-phenylpropanoic ac...)
Affinity DataEC50:  2.12E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275698((+/-)-2-(2-bromo-4-chlorophenoxy)-3-phenylpropanoi...)
Affinity DataEC50:  1.65E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275747((+/-)-2-(3,4-dichlorophenoxy)-3-phenylpropanoic ac...)
Affinity DataEC50:  4.49E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50275747((+/-)-2-(3,4-dichlorophenoxy)-3-phenylpropanoic ac...)
Affinity DataEC50:  2.55E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed