Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50027465
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50152769(CHEMBL410972 | GLP-1(7-36)-NH2 | GLP-17-(7-36) der...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275523(CHEMBL500187)
Affinity DataIC50:  5.10nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275527(CHEMBL524875)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275526(CHEMBL506368)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275522(CHEMBL525224)
Affinity DataIC50:  52nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275528(CHEMBL525608)
Affinity DataIC50:  57nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275524(CHEMBL499397)
Affinity DataIC50:  107nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275525(CHEMBL527058)
Affinity DataIC50:  113nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275523(CHEMBL500187)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275527(CHEMBL524875)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275522(CHEMBL525224)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275524(CHEMBL499397)
Affinity DataEC50:  375nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275525(CHEMBL527058)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50152769(CHEMBL410972 | GLP-1(7-36)-NH2 | GLP-17-(7-36) der...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275526(CHEMBL506368)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50275528(CHEMBL525608)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed