Compile Data Set for Download or QSAR
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Found 39 Enz. Inhib. hit(s) with all data for entry = 50041718
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413787(CHEMBL449380)
Affinity DataKi:  0.282nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413786(CHEMBL483954)
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413798(CHEMBL488149)
Affinity DataKi:  0.676nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413804(CHEMBL486171)
Affinity DataKi:  0.891nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413790(CHEMBL483969)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413791(CHEMBL483975)
Affinity DataKi:  1.62nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413816(CHEMBL516346)
Affinity DataKi:  2.19nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413797(CHEMBL488148)
Affinity DataKi:  2.24nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413817(CHEMBL473502)
Affinity DataKi:  2.51nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413803(CHEMBL487754)
Affinity DataKi:  2.82nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413789(CHEMBL521312)
Affinity DataKi:  2.82nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413806(CHEMBL486374)
Affinity DataKi:  2.95nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413807(CHEMBL516058)
Affinity DataKi:  3.63nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413802(CHEMBL488777)
Affinity DataKi:  4.27nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413799(CHEMBL487334)
Affinity DataKi:  5.62nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413794(CHEMBL390877)
Affinity DataKi:  17.4nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413808(CHEMBL474509)
Affinity DataKi:  18.2nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413818(CHEMBL474310)
Affinity DataKi:  27.5nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413819(CHEMBL474311)
Affinity DataKi:  29.5nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413805(CHEMBL486373)
Affinity DataKi:  41.7nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413795(CHEMBL488147)
Affinity DataKi:  85.1nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413812(CHEMBL475320)
Affinity DataKi:  309nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413815(CHEMBL457481)
Affinity DataKi:  347nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413813(CHEMBL513368)
Affinity DataKi:  355nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413796(CHEMBL520247)
Affinity DataKi:  417nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413814(CHEMBL472886)
Affinity DataKi:  437nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413811(CHEMBL474510)
Affinity DataKi:  513nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413823(CHEMBL514483)
Affinity DataKi:  631nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413809(CHEMBL462540)
Affinity DataKi:  871nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413810(CHEMBL500736)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413788(CHEMBL483802)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413793(CHEMBL483813)
Affinity DataKi:  2.69E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413792(CHEMBL485165)
Affinity DataKi:  3.47E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413822(CHEMBL485164)
Affinity DataKi:  3.89E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413800(CHEMBL488576)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413801(CHEMBL529896)
Affinity DataKi:  4.47E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413820(CHEMBL474917)
Affinity DataKi:  7.59E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sobhasaria Engineering College

Curated by ChEMBL
LigandPNGBDBM50413821(CHEMBL443926)
Affinity DataKi:  4.90E+4nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed