Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50027592
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50256703((1R,1aS,6aR)-4-(2-Chloro-4-trifluoromethyl-phenoxy...)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50256742(CHEMBL475053 | sodium 2-(4-((2',6'-dimethylbipheny...)
Affinity DataEC50:  260nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50256744(3-(4-(5-(thiophen-2-yl)-2,3-dihydro-1H-inden-1-ylo...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50256702(3-(4-(4-(2-(4-phenylthiazol-2-yl)-4-(pyridin-2-yl)...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50005642(1,1'-(2,4,6-trihydroxy-1,3-phenylene)bis(3-methylb...)
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHOK1 cells by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Mus musculus)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50412913(CHEMBL448569)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50256011(1,1'-(2,4,6-trihydroxy-1,3-phenylene)didodecan-1-o...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human GPR40 expressed in CHOK1 cells by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50256070(1,1'-(5-butyl-2,4,6-trihydroxy-1,3-phenylene)bis(3...)
Affinity DataEC50:  970nMAssay Description:Agonist activity at human GPR40 expressed in CHOK1 cells by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM22231((9Z,12Z)-octadeca-9,12-dienoic acid | CHEMBL267476...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human GPR40 expressed in CHOK1 cells by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM22231((9Z,12Z)-octadeca-9,12-dienoic acid | CHEMBL267476...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM22231((9Z,12Z)-octadeca-9,12-dienoic acid | CHEMBL267476...)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50005644(1,1'-(2,4,6-trihydroxy-1,3-phenylene)bis(2-methylp...)
Affinity DataEC50:  8.00E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHOK1 cells by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed