Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50027657
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50149871((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)
Affinity DataIC50:  10.2nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)
Affinity DataIC50:  11.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)
Affinity DataIC50:  11.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)
Affinity DataIC50:  20.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256745((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...)
Affinity DataIC50:  21.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)
Affinity DataIC50:  29.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)
Affinity DataIC50:  87.7nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)
Affinity DataIC50:  94.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)
Affinity DataIC50:  226nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)
Affinity DataIC50:  278nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)
Affinity DataIC50:  450nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)
Affinity DataIC50:  542nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)
Affinity DataIC50:  574nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed