Compile Data Set for Download or QSAR
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Found 141 Enz. Inhib. hit(s) with all data for entry = 50028068
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255571(4-(3-Cyano-benzenesulfonylamino)-N-[1-(2S-ethyl-4-...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255790(4-(2,4-Dimethyl-thiazole-5-sulfonylamino)-N-[1-(2S...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255627(4-(2-Cyano-benzenesulfonylamino)-N-[1-(2S-ethyl-4-...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255133(4-Benzenesulfonylamino-N-[1-(2S-ethyl-4-oxo-tetrah...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255681(CHEMBL473448 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255569(CHEMBL475669 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  1nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255570(4-(4-Cyano-benzenesulfonylamino)-N-[1-(2S-ethyl-4-...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255499(4-(4-Amino-benzenesulfonylamino)-N-[1-(2S-ethyl-4-...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255949(4-Ethanesulfonylamino-N-[1-(2S-ethyl-4-oxo-tetrahy...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255456(CHEMBL474664 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  2nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255629(CHEMBL480638 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255731(CHEMBL482218 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255680(CHEMBL480836 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255130(4-Cyclopropanesulfonylamino-N-[1-(2S-ethyl-4-oxo-t...)
Affinity DataKi:  2.40nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255849(CHEMBL471972 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255628(CHEMBL481424 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255952(CHEMBL482348 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255500(CHEMBL475269 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255950(4-(Butane-1-sulfonylamino)-N-[1-(2S-ethyl-4-oxo-te...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255457(CHEMBL474865 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255458(CHEMBL515588 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255498(CHEMBL475063 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255354(4-Benzenesulfonylamino-N-[1-(2S-ethyl-4-oxo-tetrah...)
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255732(CHEMBL519136 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255297(CHEMBL479461 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255132(4-(N-Dimethylamino)-sulfonylamino-N-[1-(2S-ethyl-4...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255351(3-Chloro-N-[1-(2S-ethyl-4-oxo-tetrahydro-furan-3S-...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255789(CHEMBL474257 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255682(4-(2-Chloro-pyridine-3-sulfonylamino)-N-[1-(2S-eth...)
Affinity DataKi:  5.90nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255951(CHEMBL519633 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  8.30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255791(CHEMBL481986 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  8.60nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255408(4-Benzenesulfonylamino-3-chloro-N-[1-(2S-ethyl-4-o...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255894(CHEMBL481503 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255733(CHEMBL481433 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255352(CHEMBL481034 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255295(CHEMBL480634 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  26nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255298(CHEMBL516749 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255848(CHEMBL512367 | N-((S)-1-((2S,3S)-2-ethyl-4-oxotetr...)
Affinity DataKi:  31nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255176(CHEMBL475062 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  31nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255409(6-Benzenesulfonylamino-N-[1-(2S-ethyl-4-oxo-tetrah...)
Affinity DataKi:  56nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255353(3-Acetyl-N-[1-(2S-ethyl-4-oxo-tetrahydro-furan-3S-...)
Affinity DataKi:  57nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255410(CHEMBL519763 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  63nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255895(CHEMBL482166 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  98nMAssay Description:Inhibition of human recombinant cathepsin K expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255895(CHEMBL482166 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255896(CHEMBL482167 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  140nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255131(4-Cyclohexanesulfonylamino-N-[1-(2S-ethyl-4-oxotet...)
Affinity DataKi:  180nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255897(CHEMBL482168 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255297(CHEMBL479461 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  240nMAssay Description:Inhibition of human recombinant cathepsin K expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255681(CHEMBL473448 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  260nMAssay Description:Inhibition of human recombinant cathepsin K expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255569(CHEMBL475669 | N-[1-(2S-Ethyl-4-oxo-tetrahydro-fur...)
Affinity DataKi:  270nMAssay Description:Inhibition of human recombinant cathepsin K expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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