Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50038805
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267023(1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-5-(4-ethylphen...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267025(1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-3-hydroxy-5-(4...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267024(1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-5-(4-ethoxyphe...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267053(1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-3-hydroxy-5-(4...)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM2681(3-{1-[3-(dimethylamino)propyl]-1H-indol-3-yl}-4-(1...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267091(BAS-1059623 | CHEMBL476454 | N-(2-(1H-indol-3-yl)e...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267089(2-morpholino-8-phenylchroman-4-one | CHEMBL476452 ...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267090(2-(3-(9H-carbazol-9-yl)-2-hydroxypropoxy)benzaldeh...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed