Compile Data Set for Download or QSAR
maximum 50k data
Found 320 Enz. Inhib. hit(s) with all data for entry = 50028244
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of ErbB2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248349(CHEMBL473553 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  63nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248413(CHEMBL491686 | N2-(3-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  100nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248293(CHEMBL473556 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  135nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248413(CHEMBL491686 | N2-(3-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  160nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248413(CHEMBL491686 | N2-(3-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248294(CHEMBL514942 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  240nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  280nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248229(CHEMBL474347 | N-(4-(benzo[d]thiazol-2-yl)-2-fluor...)
Affinity DataIC50:  290nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248292(CHEMBL473354 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  310nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248147(CHEMBL461110 | N2-(4-(benzo[d]thiazol-2-yl)-3-meth...)
Affinity DataIC50:  320nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248293(CHEMBL473556 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248146(CHEMBL461109 | N2-(4-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  480nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248232(CHEMBL514016 | N-(4-(benzo[d]thiazol-2-yl)-3-chlor...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(CHEMBL473557 | N-(4-(benzo[d]thiazol-2-yl)-2-fluor...)
Affinity DataIC50:  510nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  510nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248232(CHEMBL514016 | N-(4-(benzo[d]thiazol-2-yl)-3-chlor...)
Affinity DataIC50:  600nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  610nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248350(CHEMBL514941 | N4-(4-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  630nMAssay Description:Inhibition of insulin receptor by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248230(CHEMBL474543 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  630nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248230(CHEMBL474543 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  640nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  700nMAssay Description:Inhibition of CDK2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(CHEMBL473557 | N-(4-(benzo[d]thiazol-2-yl)-2-fluor...)
Affinity DataIC50:  700nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248185(CHEMBL472946 | N-(4-(benzo[d]thiazol-2-yl)phenyl)t...)
Affinity DataIC50:  720nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248149(CHEMBL462162 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  720nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248230(CHEMBL474543 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  750nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248414(CHEMBL522785 | N4-(3-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  780nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248232(CHEMBL514016 | N-(4-(benzo[d]thiazol-2-yl)-3-chlor...)
Affinity DataIC50:  800nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248232(CHEMBL514016 | N-(4-(benzo[d]thiazol-2-yl)-3-chlor...)
Affinity DataIC50:  800nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(CHEMBL473557 | N-(4-(benzo[d]thiazol-2-yl)-2-fluor...)
Affinity DataIC50:  800nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248232(CHEMBL514016 | N-(4-(benzo[d]thiazol-2-yl)-3-chlor...)
Affinity DataIC50:  800nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248414(CHEMBL522785 | N4-(3-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  810nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248416(CHEMBL443906 | N-(3-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  840nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248120(CHEMBL459886 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  840nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248294(CHEMBL514942 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  840nMAssay Description:Inhibition of TIE2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248230(CHEMBL474543 | N-(4-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  860nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248416(CHEMBL443906 | N-(3-(benzo[d]thiazol-2-yl)phenyl)-...)
Affinity DataIC50:  870nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  900nMAssay Description:Inhibition of FAK by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  900nMAssay Description:Inhibition of insulin receptor by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248464(CHEMBL491677 | N-[4-(isoindolin-2-yl)phenyl]-6',7'...)
Affinity DataIC50:  920nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248414(CHEMBL522785 | N4-(3-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  940nMAssay Description:Inhibition of insulin receptor by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  960nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248414(CHEMBL522785 | N4-(3-(benzo[d]thiazol-2-yl)phenyl)...)
Affinity DataIC50:  960nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(CHEMBL473557 | N-(4-(benzo[d]thiazol-2-yl)-2-fluor...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(CHEMBL473557 | N-(4-(benzo[d]thiazol-2-yl)-2-fluor...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of TIE2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(CHEMBL460746 | N-(3-(benzo[d]thiazol-2-yl)-4-hydro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of VEGFR3 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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