Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50030410
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295778(2-(2,6-dimethylphenoxy)-5-(4-(6-methoxypyridin-3-y...)
Affinity DataKi:  5.90nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295779(2-(2-chloro-3,6-difluorophenoxy)-5-(4-(6-methoxypy...)
Affinity DataKi:  8.80nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295777(2-(4-fluoro-2-methylphenoxy)-5-(4-(6-methoxypyridi...)
Affinity DataKi:  9.40nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295772(2-(4-(6-methoxypyridin-3-yl)-5-methyl-4H-1,2,4-tri...)
Affinity DataKi:  12.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295776(2-(3-fluoro-2-methylphenoxy)-5-(4-(6-methoxypyridi...)
Affinity DataKi:  14.6nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295771(2-(2-chlorophenoxy)-5-(4-(6-methoxypyridin-3-yl)-5...)
Affinity DataKi:  23.6nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295780(2-(2,4-dichlorophenoxy)-5-(4-(6-methoxypyridin-3-y...)
Affinity DataKi:  37.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295773(2-(2-ethylphenoxy)-5-(4-(6-methoxypyridin-3-yl)-5-...)
Affinity DataKi:  52.3nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295775(2-(4-(6-methoxypyridin-3-yl)-5-methyl-4H-1,2,4-tri...)
Affinity DataKi:  198nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295774(2-(2-methoxyphenoxy)-5-(4-(6-methoxypyridin-3-yl)-...)
Affinity DataKi:  253nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295770(2-(4-(6-methoxypyridin-3-yl)-5-methyl-4H-1,2,4-tri...)
Affinity DataKi:  350nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  388nMAssay Description:Antagonist activity at human cloned vasopressin V1A receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295770(2-(4-(6-methoxypyridin-3-yl)-5-methyl-4H-1,2,4-tri...)
Affinity DataKi:  2.32E+3nMAssay Description:Antagonist activity at human cloned vasopressin V1A receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295770(2-(4-(6-methoxypyridin-3-yl)-5-methyl-4H-1,2,4-tri...)
Affinity DataKi:  2.32E+3nMAssay Description:Antagonist activity at human cloned vasopressin V1A receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed