Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50028657
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]PDBu form human PKCbeta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]PDBu form human PKCalpha in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  268nMAssay Description:Displacement of [3H]PDBu form human PKCepsilon in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed