Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50028786
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268759(CHEMBL496032 | N-butyl-2-chloro-N-(2-(4-(4-chlorop...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268683(CHEMBL496812 | N-butyl-2-chloro-N-(2-(4-(4-methoxy...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268633(CHEMBL498425 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268634(CHEMBL498627 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268514(CHEMBL522247 | N-butyl-2-chloro-N-(2-(4-(4-methoxy...)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268758(CHEMBL495836 | N-butyl-2-chloro-N-(2-(4-(4-fluorop...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268632(CHEMBL498424 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268454(2-chloro-N-isopropyl-N-(2-(4-(4-methoxyphenyl)pyrr...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268569(CHEMBL496596 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  236nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268721(CHEMBL496221 | N-butyl-2-chloro-N-(2-oxo-2-(4-phen...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268568(CHEMBL521738 | N-butyl-2-fluoro-N-(2-(4-(4-methoxy...)
Affinity DataKi:  349nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268682(CHEMBL496207 | N-butyl-2-methoxy-N-(2-(4-(4-methox...)
Affinity DataKi:  461nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268567(CHEMBL497006 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  503nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268681(CHEMBL521717 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  539nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268570(CHEMBL496597 | N-butyl-N-(2-(4-(4-methoxyphenyl)py...)
Affinity DataKi:  602nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50268513(CHEMBL526749 | N-butyl-3,5-dichloro-N-(2-(4-(4-met...)
Affinity DataKi:  831nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed