Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50028793
TargetDynamin-1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50268295(2-Cyano-N-octyl-3-(1-(3-dimethylaminopropyl)-1H-in...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of dynamin 1-mediated endocytosis internalization of Tf-A594 in human U2OS cells pretreated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDynamin-1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50268962(2-Cyano-N-octyl-3-[1-(3-dimethylaminopropyl)-2-met...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of dynamin 1-mediated endocytosis internalization of Tf-A594 in human U2OS cells pretreated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDynamin-1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50268872(2-Cyano-N-octyl-3-[1-(2-dimethylaminoethyl)-2-meth...)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of dynamin 1-mediated endocytosis internalization of Tf-A594 in human U2OS cells pretreated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDynamin-1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50268961(2-Cyano-N-hexyl-3-[1-(3-dimethylaminopropyl)-2-met...)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of dynamin 1-mediated endocytosis internalization of Tf-A594 in human U2OS cells pretreated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDynamin-1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50268963(2-Cyano-N-decyl-3-[1-(2-dimethylaminoethyl)-2-meth...)
Affinity DataIC50:  5.82E+4nMAssay Description:Inhibition of dynamin 1-mediated endocytosis internalization of Tf-A594 in human U2OS cells pretreated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed