Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50030418
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50295871(CHEMBL552002 | N-[2-(5-Methoxy-2-{[(4-methoxypheny...)
Affinity DataKi:  8nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50295871(CHEMBL552002 | N-[2-(5-Methoxy-2-{[(4-methoxypheny...)
Affinity DataKi:  9nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50295870(CHEMBL563847 | N-{2-(5-Methoxy-2-({[methyl[4-(trif...)
Affinity DataKi:  63nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50295870(CHEMBL563847 | N-{2-(5-Methoxy-2-({[methyl[4-(trif...)
Affinity DataKi:  111nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50273283(CHEMBL455909 | N-[2-(13a,14-Dihydro-6H,13H-pyrazin...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50273283(CHEMBL455909 | N-[2-(13a,14-Dihydro-6H,13H-pyrazin...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50295869(CHEMBL556908 | N-[2-(8-Methoxy-2-methyl-1,2,3,4-te...)
Affinity DataIC50:  3.14nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed