Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50030767
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301066(CHEMBL571939 | N-(6-(2-(((2S,3S,4R,5R)-3,4-dihydro...)
Affinity DataKi:  0.0180nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in HL60 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301067(CHEMBL569223 | N-(6-(2-(((2S,3S,4R,5R)-3,4-dihydro...)
Affinity DataKi:  0.0640nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in HL60 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301066(CHEMBL571939 | N-(6-(2-(((2S,3S,4R,5R)-3,4-dihydro...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in HL60 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301067(CHEMBL569223 | N-(6-(2-(((2S,3S,4R,5R)-3,4-dihydro...)
Affinity DataIC50:  5.10nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in HL60 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301068(5'-[(fluorescein-5-ylcarbonyl)-6-aminohexanoyl-(2-...)
Affinity DataKd:  0.360nMAssay Description:Binding affinity to human ENT1 in BX-PC3 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301068(5'-[(fluorescein-5-ylcarbonyl)-6-aminohexanoyl-(2-...)
Affinity DataKd:  0.910nMAssay Description:Binding affinity to human ENT1 in MIA-PaCa2 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301068(5'-[(fluorescein-5-ylcarbonyl)-6-aminohexanoyl-(2-...)
Affinity DataKd:  3.80nMAssay Description:Binding affinity to human ENT1 in panc1 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301068(5'-[(fluorescein-5-ylcarbonyl)-6-aminohexanoyl-(2-...)
Affinity DataKd:  0.320nMAssay Description:Binding affinity to human ENT1 in Capan1 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301068(5'-[(fluorescein-5-ylcarbonyl)-6-aminohexanoyl-(2-...)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to human ENT1 in SK-PC1 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Ulm University

Curated by ChEMBL
LigandPNGBDBM50301068(5'-[(fluorescein-5-ylcarbonyl)-6-aminohexanoyl-(2-...)
Affinity DataKd:  0.260nMAssay Description:Binding affinity to human ENT1 in HL60 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed