Compile Data Set for Download or QSAR
maximum 50k data
Found 80 Enz. Inhib. hit(s) with all data for entry = 50041771
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415167(CHEMBL606753)
Affinity DataKi:  7.41nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415168(CHEMBL593217)
Affinity DataKi:  12.9nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415169(CHEMBL594271)
Affinity DataKi:  13.8nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415171(CHEMBL595658)
Affinity DataKi:  14.8nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415173(CHEMBL594734)
Affinity DataKi:  19.1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415191(CHEMBL603209)
Affinity DataKi:  21.4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415172(CHEMBL594735)
Affinity DataKi:  21.4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415181(CHEMBL596346)
Affinity DataKi:  26.9nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415183(CHEMBL593572)
Affinity DataKi:  27.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415168(CHEMBL593217)
Affinity DataKi:  28.8nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415170(CHEMBL604075)
Affinity DataKi:  32.4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415180(CHEMBL594963)
Affinity DataKi:  35.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415179(CHEMBL603861)
Affinity DataKi:  38.9nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415181(CHEMBL596346)
Affinity DataKi:  43.6nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415189(CHEMBL595657)
Affinity DataKi:  46.8nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415185(CHEMBL606535)
Affinity DataKi:  61.7nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415167(CHEMBL606753)
Affinity DataKi:  83.2nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by microplate beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415184(CHEMBL604885)
Affinity DataKi:  89.1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415178(CHEMBL594728)
Affinity DataKi:  89.1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415168(CHEMBL593217)
Affinity DataKi:  89.1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by microplate beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415184(CHEMBL604885)
Affinity DataKi:  89.1nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415190(CHEMBL604492)
Affinity DataKi:  93.3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415180(CHEMBL594963)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415167(CHEMBL606753)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415169(CHEMBL594271)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by microplate beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415169(CHEMBL594271)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415175(CHEMBL596558)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415189(CHEMBL595657)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415174(CHEMBL595431)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415182(CHEMBL604896)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415191(CHEMBL603209)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415173(CHEMBL594734)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415172(CHEMBL594735)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415170(CHEMBL604075)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by microplate beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415190(CHEMBL604492)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415186(CHEMBL594255)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415185(CHEMBL606535)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415171(CHEMBL595658)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415179(CHEMBL603861)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415187(CHEMBL596125)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415187(CHEMBL596125)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415177(CHEMBL604283)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415171(CHEMBL595658)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by microplate beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415177(CHEMBL604283)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415192(CHEMBL594970)
Affinity DataKi:  275nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415175(CHEMBL596558)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415173(CHEMBL594734)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by microplate beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415172(CHEMBL594735)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by microplate beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415176(CHEMBL593216)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50415194(CHEMBL596331)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]DPCPX form adenosine A1 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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