Compile Data Set for Download or QSAR
maximum 50k data
Found 50 Enz. Inhib. hit(s) with all data for entry = 50030732
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300648(4-(3-((S)-1-((cis)-2-((S)-5-amino-1-(benzylamino)-...)
Affinity DataIC50:  68nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300657(4-(3-((S)-1-((cis)-2-((2R,3S)-6-amino-2-(benzyloxy...)
Affinity DataIC50:  69nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300658(4-((E)-3-((S)-1-((1R,2S,5S)-2-(2-(benzyloxy)ethylc...)
Affinity DataIC50:  69nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300656(4-(3-((S)-1-((cis)-2-((S)-5-amino-1-(benzyloxy)-5-...)
Affinity DataIC50:  94nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300627(4-(3-((S)-1-((S)-2-((R)-5-amino-5-oxopentan-2-ylca...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300646(4-(3-((S)-4-methyl-1-oxo-1-((S)-2-(2-ureidoethylca...)
Affinity DataIC50:  131nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50198780(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(benzylamino)-1,...)
Affinity DataIC50:  138nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300650(4-(3-((S)-1-((cis)-2-((R)-5-amino-5-oxopentan-2-yl...)
Affinity DataIC50:  175nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300634(4-(3-((S)-1-((S)-2-((2R,3S)-6-amino-2-(benzyloxy)-...)
Affinity DataIC50:  272nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50423685(CHEMBL502473)
Affinity DataIC50:  290nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300655((S)-5-amino-2-((cis)-3-((S)-4-methyl-2-(3-(4-(phos...)
Affinity DataIC50:  290nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300633(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(benzyloxy)-5-ox...)
Affinity DataIC50:  294nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300649(4-(3-((S)-1-((cis)-2-(4-amino-4-oxobutylcarbamoyl)...)
Affinity DataIC50:  303nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300642(2-((S)-1-((S)-4-methyl-2-(3-(4-(phosphonooxy)pheny...)
Affinity DataIC50:  360nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50198778((S)-3-(benzylamino)-2-((S)-1-((S)-4-methyl-2-(3-(4...)
Affinity DataIC50:  379nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300654(4-(3-((S)-1-((cis)-2-((2R,3S)-6-amino-2-hydroxy-6-...)
Affinity DataIC50:  437nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300644((R)-3-(benzyloxy)-2-((S)-1-((S)-4-methyl-2-(3-(4-(...)
Affinity DataIC50:  454nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300653(4-(3-((S)-1-((cis)-2-((R)-1-amino-1-oxooctan-4-ylc...)
Affinity DataIC50:  499nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300651(4-(3-((S)-1-((cis)-2-((S)-6-amino-2-methyl-6-oxohe...)
Affinity DataIC50:  511nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300618(4-(3-((S)-1-((S)-2-(4-amino-4-oxobutylcarbamoyl)py...)
Affinity DataIC50:  574nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300641(4-(3-((S)-1-((S)-2-((S)-1-acetamido-5-amino-5-oxop...)
Affinity DataIC50:  589nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300635((S)-5-amino-2-((S)-1-((S)-4-methyl-2-(3-(4-(phosph...)
Affinity DataIC50:  615nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300643((R)-2-((S)-1-((S)-4-methyl-2-(3-(4-(phosphonooxy)p...)
Affinity DataIC50:  797nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300632(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(4-hydroxyphenyl...)
Affinity DataIC50:  848nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50198779((2R,3S)-4-(benzylamino)-3-((S)-1-((S)-4-methyl-2-(...)
Affinity DataIC50:  850nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300614(4-(3-((S)-1-((S)-2-((S)-4-amino-1-(benzylamino)-1,...)
Affinity DataIC50:  874nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300639(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(dibenzylamino)-...)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300619(4-(3-((S)-1-((S)-2-((E)-4-amino-4-oxobut-2-enylcar...)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300620(4-(3-((S)-1-((S)-2-(4-amino-4-oxobut-2-ynylcarbamo...)
Affinity DataIC50:  1.14E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300628(4-(3-((S)-1-((S)-2-((S)-5-amino-5-oxopentan-2-ylca...)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300636(4-(3-((S)-1-((S)-2-((S)-5-amino-5-oxo-1-(piperidin...)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300640((S)-5-amino-2-((S)-1-((S)-4-methyl-2-(3-(4-(phosph...)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300637(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(4-methylpiperaz...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300631(4-(3-((S)-1-((S)-2-((R)-1-amino-1-oxooctan-4-ylcar...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300647(4-(3-((S)-4-methyl-1-oxo-1-((S)-2-((R)-1-ureidopro...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300615(4-(3-((S)-1-((S)-2-((S)-6-amino-1-(benzylamino)-1,...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300638(4-(3-((S)-1-((S)-2-((S)-5-amino-1-morpholino-5-oxo...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300652(4-(3-((S)-1-((cis)-2-((S)-1-amino-6-methyl-1-oxohe...)
Affinity DataIC50:  1.63E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300626(4-(3-((S)-1-((S)-2-(4-hydrazinyl-4-oxobutylcarbamo...)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300629(4-(3-((S)-1-((S)-2-((S)-6-amino-2-methyl-6-oxohexa...)
Affinity DataIC50:  1.88E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300625(4-(3-((S)-1-((S)-2-(4-(hydroxyamino)-4-oxobutylcar...)
Affinity DataIC50:  2.64E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300622(4-(3-((S)-1-((S)-2-((3S,5S)-5-carbamoylpyrrolidin-...)
Affinity DataIC50:  3.21E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300621(4-(3-((S)-1-((S)-2-((S)-2-(3-amino-3-oxopropyl)pyr...)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300623(4-(3-((S)-1-((S)-2-((3R,5S)-5-carbamoylpyrrolidin-...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300630(4-(3-((S)-1-((S)-2-((S)-1-amino-6-methyl-1-oxohept...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300613(4-(3-((S)-1-((S)-2-(2-(benzylamino)-2-oxoethylcarb...)
Affinity DataIC50:  4.94E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300645((2S,3R)-3-(benzyloxy)-2-((S)-1-((S)-4-methyl-2-(3-...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300617(4-(3-((S)-1-((S)-2-((S)-1-amino-1-oxopropan-2-ylca...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300616(4-(3-((S)-1-((S)-2-carbamoylpyrrolidin-1-yl)-4-met...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50300624(4-(3-((S)-4-methyl-1-oxo-1-((S)-2-(3-sulfamoylprop...)
Affinity DataIC50:  6.82E+4nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed