Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50030835
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)
Affinity DataIC50:  500nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant PI3Kdelta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302392(6-methoxy-3-(5-(3-methoxyphenyl)-1,2,4-oxadiazol-3...)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant PI3Kdelta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant PI3Kbeta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302392(6-methoxy-3-(5-(3-methoxyphenyl)-1,2,4-oxadiazol-3...)
Affinity DataIC50:  900nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302392(6-methoxy-3-(5-(3-methoxyphenyl)-1,2,4-oxadiazol-3...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human recombinant PI3Kbeta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302389(3-(benzo[d]thiazol-2-yl)-7-hydroxy-2H-chromen-2-on...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302389(3-(benzo[d]thiazol-2-yl)-7-hydroxy-2H-chromen-2-on...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of recombinant PI3Kdelta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302393(3-(6-chloro-2-oxobenzo[d]oxazol-3(2H)-yl)-N-phenyl...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human recombinant PI3Kbeta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302389(3-(benzo[d]thiazol-2-yl)-7-hydroxy-2H-chromen-2-on...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human recombinant PI3Kbeta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302393(3-(6-chloro-2-oxobenzo[d]oxazol-3(2H)-yl)-N-phenyl...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302391(1,7-dimethyl-1H-pyrazolo[3,4-b]quinolin-3-yl 2-phe...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302391(1,7-dimethyl-1H-pyrazolo[3,4-b]quinolin-3-yl 2-phe...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of recombinant PI3Kdelta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302394(3-(2-methoxy-6-phenylpyridin-3-yl)-5-(pyridin-4-yl...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302390(CHEMBL579219 | methyl 5-((5,6-dimethylthieno[2,3-d...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant PI3Kdelta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302394(3-(2-methoxy-6-phenylpyridin-3-yl)-5-(pyridin-4-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant PI3Kbeta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302395(3-(5-(2-methoxyphenyl)-1,2,4-oxadiazol-3-yl)-6-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302390(CHEMBL579219 | methyl 5-((5,6-dimethylthieno[2,3-d...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant PI3Kbeta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302391(1,7-dimethyl-1H-pyrazolo[3,4-b]quinolin-3-yl 2-phe...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant PI3Kbeta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Mus musculus (Mouse))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302390(CHEMBL579219 | methyl 5-((5,6-dimethylthieno[2,3-d...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse recombinant PI3Kalpha expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50302393(3-(6-chloro-2-oxobenzo[d]oxazol-3(2H)-yl)-N-phenyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant PI3Kdelta expressed in baculovirus-infected Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed