Compile Data Set for Download or QSAR
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Found 93 Enz. Inhib. hit(s) with all data for entry = 50030742
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268555(6-(3-(furan-3-yl)benzylamino)-9-(3-hydroxypropyl)-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300772(6-(3-(1H-indol-5-yl)benzylamino)-9-(3-hydroxypropy...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268557(9-(3-hydroxypropyl)-6-(3-(thiophen-3-yl)benzylamin...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268616(9-(3-hydroxypropyl)-6-(3-(pyridin-3-yl)benzylamino...)
Affinity DataIC50:  260nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50300773(6-(3-(1H-indol-6-yl)benzylamino)-9-(3-hydroxypropy...)
Affinity DataIC50:  260nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268554(6-(3-(furan-2-yl)benzylamino)-9-(3-hydroxypropyl)-...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50300774(CHEMBL570364 | N-(3'-((2-cyano-9-(3-hydroxypropyl)...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300774(CHEMBL570364 | N-(3'-((2-cyano-9-(3-hydroxypropyl)...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300773(6-(3-(1H-indol-6-yl)benzylamino)-9-(3-hydroxypropy...)
Affinity DataIC50:  460nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268557(9-(3-hydroxypropyl)-6-(3-(thiophen-3-yl)benzylamin...)
Affinity DataIC50:  480nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268446(CHEMBL496404 | methyl 3'-((2-cyano-9-(3-hydroxypro...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50300772(6-(3-(1H-indol-5-yl)benzylamino)-9-(3-hydroxypropy...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268555(6-(3-(furan-3-yl)benzylamino)-9-(3-hydroxypropyl)-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268553(9-(3-hydroxypropyl)-6-(3-(naphthalen-2-yl)benzylam...)
Affinity DataIC50:  700nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300781(6-((3'-chlorobiphenyl-3-yl)methylamino)-9-(3-hydro...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268668(6-(biphenyl-3-ylmethylamino)-9-(3-hydroxypropyl)-9...)
Affinity DataIC50:  700nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268553(9-(3-hydroxypropyl)-6-(3-(naphthalen-2-yl)benzylam...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268500(1-butyl-4-(2-(4'-ethylbiphenyl-3-yl)ethyl)-6-ethyn...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268446(CHEMBL496404 | methyl 3'-((2-cyano-9-(3-hydroxypro...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268556(9-(3-hydroxypropyl)-6-(3-(thiophen-2-yl)benzylamin...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268668(6-(biphenyl-3-ylmethylamino)-9-(3-hydroxypropyl)-9...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268554(6-(3-(furan-2-yl)benzylamino)-9-(3-hydroxypropyl)-...)
Affinity DataIC50:  840nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50258405(6-((3',4'-dichlorobiphenyl-3-yl)methylamino)-9-(3-...)
Affinity DataIC50:  900nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268444(6-((3'-(dimethylamino)biphenyl-3-yl)methylamino)-9...)
Affinity DataIC50:  900nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50258404(6-((3',5'-dichlorobiphenyl-3-yl)methylamino)-9-(3-...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268556(9-(3-hydroxypropyl)-6-(3-(thiophen-2-yl)benzylamin...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300779(9-(3-hydroxypropyl)-6-((2'-isopropylbiphenyl-3-yl)...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300784(9-(3-hydroxypropyl)-6-(3-(1-(phenylsulfonyl)-1H-in...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300778(6-((2',6'-dimethylbiphenyl-3-yl)methylamino)-9-(3-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268502(9-(3-hydroxypropyl)-6-((4'-vinylbiphenyl-3-yl)meth...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268500(1-butyl-4-(2-(4'-ethylbiphenyl-3-yl)ethyl)-6-ethyn...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268670(9-(3-hydroxypropyl)-6-((2'-methylbiphenyl-3-yl)met...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50258404(6-((3',5'-dichlorobiphenyl-3-yl)methylamino)-9-(3-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50300781(6-((3'-chlorobiphenyl-3-yl)methylamino)-9-(3-hydro...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50300782(CHEMBL571938 | methyl 3'-((2-cyano-9-(3-hydroxypro...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268620(6-((3'-bromo-2'-isopropoxybiphenyl-3-yl)methylamin...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268445(6-((4'-chlorobiphenyl-3-yl)methylamino)-9-(3-hydro...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268444(6-((3'-(dimethylamino)biphenyl-3-yl)methylamino)-9...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300780(CHEMBL571276 | methyl 3'-((2-cyano-9-(3-hydroxypro...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268501(9-(3-hydroxypropyl)-6-((3'-vinylbiphenyl-3-yl)meth...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300785(9-(3-hydroxypropyl)-6-((2'-(trifluoromethyl)biphen...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268501(9-(3-hydroxypropyl)-6-((3'-vinylbiphenyl-3-yl)meth...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268620(6-((3'-bromo-2'-isopropoxybiphenyl-3-yl)methylamin...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268616(9-(3-hydroxypropyl)-6-(3-(pyridin-3-yl)benzylamino...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50258405(6-((3',4'-dichlorobiphenyl-3-yl)methylamino)-9-(3-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300782(CHEMBL571938 | methyl 3'-((2-cyano-9-(3-hydroxypro...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50268502(9-(3-hydroxypropyl)-6-((4'-vinylbiphenyl-3-yl)meth...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50300783(9-(3-hydroxypropyl)-6-(3-(1-(phenylsulfonyl)-1H-in...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50268445(6-((4'-chlorobiphenyl-3-yl)methylamino)-9-(3-hydro...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human liver cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50300784(9-(3-hydroxypropyl)-6-(3-(1-(phenylsulfonyl)-1H-in...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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