Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50030518
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297420((Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  2.01nMAssay Description:Inhibition of [3H]serotonin reuptake at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297420((Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of [3H]serotonin reuptake at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297420((Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  4.16nMAssay Description:Inhibition of [3H]norepinephrine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297420((Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  4.16nMAssay Description:Inhibition of [3H]norepinephrine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataKi:  5.07nMAssay Description:Inhibition of [3H]dopamine reuptake at dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  5.11nMAssay Description:Inhibition of [3H]norepinephrine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297418((E)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  7.47nMAssay Description:Inhibition of [3H]serotonin reuptake at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297418((E)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  7.47nMAssay Description:Inhibition of [3H]serotonin reuptake at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  7.57nMAssay Description:Inhibition of [3H]serotonin reuptake at serotonin transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297421(CHEMBL558525 | N-methyl-1-((1R,2R)-2-(naphthalen-1...)
Affinity DataKi:  27.8nMAssay Description:Inhibition of [3H]norepinephrine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297421(CHEMBL558525 | N-methyl-1-((1R,2R)-2-(naphthalen-1...)
Affinity DataKi:  30.4nMAssay Description:Inhibition of [3H]serotonin reuptake at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297419(CHEMBL558065 | N-methyl-1-((1S,2R)-2-(naphthalen-1...)
Affinity DataKi:  33.2nMAssay Description:Inhibition of [3H]serotonin reuptake at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297418((E)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  75.7nMAssay Description:Inhibition of [3H]norepinephrine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297418((E)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  75.7nMAssay Description:Inhibition of [3H]norepinephrine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297419(CHEMBL558065 | N-methyl-1-((1S,2R)-2-(naphthalen-1...)
Affinity DataKi:  153nMAssay Description:Inhibition of [3H]norepinephrine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297420((Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  283nMAssay Description:Inhibition of [3H]dopamine reuptake at dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297420((Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  283nMAssay Description:Inhibition of [3H]dopamine reuptake at dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297418((E)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  586nMAssay Description:Inhibition of [3H]dopamine reuptake at dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297418((E)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-...)
Affinity DataKi:  586nMAssay Description:Inhibition of [3H]dopamine reuptake at dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297419(CHEMBL558065 | N-methyl-1-((1S,2R)-2-(naphthalen-1...)
Affinity DataKi:  913nMAssay Description:Inhibition of [3H]dopamine reuptake at dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50297421(CHEMBL558525 | N-methyl-1-((1R,2R)-2-(naphthalen-1...)
Affinity DataKi:  1.91E+3nMAssay Description:Inhibition of [3H]dopamine reuptake at dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed