TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Binding affinity to LPA3More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 5(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 292nMAssay Description:Binding affinity to LPA5More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 311nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 1.08E+3nMAssay Description:Binding affinity to LPA3More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Antagonist activity at LPA1 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Antagonist activity at LPA1 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 355nMAssay Description:Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 5(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 463nMAssay Description:Antagonist activity at LPA5 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 609nMAssay Description:Antagonist activity at LPA1 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 752nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 2.99E+3nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 2.74E+4nMAssay Description:Antagonist activity at LPA1 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair