Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50030645
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299557((S)-2-((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataKi:  0.248nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299558(CHEMBL583488 | H-4'-carboxamido-2',6'-dimethylphen...)
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299559(CHEMBL583285 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  0.536nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299560(CHEMBL572542 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  0.605nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299561(CHEMBL572543 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  0.646nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299562(CHEMBL572494 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  0.783nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299563(CHEMBL583487 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  0.825nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  1.22nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi:  1.84nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299566(CHEMBL583485 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299567(CHEMBL583486 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  3.31nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299560(CHEMBL572542 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  87.7nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299557((S)-2-((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299562(CHEMBL572494 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299559(CHEMBL583285 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50060080(2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299560(CHEMBL572542 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299566(CHEMBL583485 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  323nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299567(CHEMBL583486 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  334nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299562(CHEMBL572494 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  597nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299563(CHEMBL583487 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  615nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299558(CHEMBL583488 | H-4'-carboxamido-2',6'-dimethylphen...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299557((S)-2-((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50060080(2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299566(CHEMBL583485 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299559(CHEMBL583285 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299567(CHEMBL583486 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299558(CHEMBL583488 | H-4'-carboxamido-2',6'-dimethylphen...)
Affinity DataKi:  2.21E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299561(CHEMBL572543 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299563(CHEMBL583487 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  2.75E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299561(CHEMBL572543 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  4.76E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50060080(2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299560(CHEMBL572542 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataIC50:  3.42nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as effect on muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299557((S)-2-((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataIC50:  769nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as effect on muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as effect on muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed