Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50031348
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM27641(1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-[(...)
Affinity DataIC50:  60nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311688(CHEMBL1080460 | N-(2-methoxybenzyl)-1-(3-((2-(meth...)
Affinity DataIC50:  200nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311707(1-(3-((2-(methylamino)ethylamino)methyl)phenyl)-N-...)
Affinity DataIC50:  320nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311700(CHEMBL1087114 | N-(5-fluoro-2-methoxybenzyl)-1-(3-...)
Affinity DataIC50:  710nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311699(CHEMBL1087540 | N-((2,3-dihydrobenzo[b][1,4]dioxin...)
Affinity DataIC50:  710nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311698(CHEMBL1088320 | N-(2-ethoxybenzyl)-1-(3-((2-(methy...)
Affinity DataIC50:  900nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311689(1-(3-((2-aminoethylamino)methyl)phenyl)-N-(2-metho...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311697(CHEMBL1088188 | N-(2-ethylbenzyl)-1-(3-((2-(methyl...)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311706(CHEMBL1087878 | N-(2-(1H-indol-3-yl)ethyl)-1-(3-((...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311708(CHEMBL1080335 | N-((2-methoxynaphthalen-1-yl)methy...)
Affinity DataIC50:  3.35E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311703(CHEMBL1088567 | N-(cyclohexylmethyl)-1-(3-((2-(met...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311705(CHEMBL1087877 | N-((1H-benzo[d]imidazol-2-yl)methy...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311684((S)-1-(3-((2-aminopropanethioamido)methyl)phenyl)-...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311704(CHEMBL1088568 | N-((1-methyl-1H-benzo[d]imidazol-2...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311709(1-(4-fluoro-3-((2-(methylamino)ethylamino)methyl)p...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311701(1-(3-((2-(methylamino)ethylamino)methyl)phenyl)-N-...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311691(1-(3-((2-(ethylamino)ethylamino)methyl)phenyl)-N-(...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311690(1-(3-((2-(dimethylamino)ethylamino)methyl)phenyl)-...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311710(CHEMBL1080519 | N-(2-methoxybenzyl)-1-(4-methyl-3-...)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311702(CHEMBL1087234 | N-(2-aminobenzyl)-1-(3-((2-(methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311695(CHEMBL1086763 | N-benzyl-1-(3-((2-(methylamino)eth...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311712(5-(2-methoxybenzyl)-8-((2-(methylamino)ethylamino)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311696(1-(3-((2-(methylamino)ethylamino)methyl)phenyl)-N-...)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311694(CHEMBL1080477 | N-(2-methoxybenzyl)-1-(3-(2-(methy...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311692(CHEMBL1080125 | N-(2-methoxybenzyl)-1-(3-((pyrroli...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311687((S)-1-(3-(5-(1-aminoethyl)-1,2,4-oxadiazol-3-yl)ph...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311686((S)-1-(3-(5-(1-aminoethyl)-1H-1,2,4-triazol-3-yl)p...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311685((S)-1-(3-((2-hydroxypropanamido)methyl)phenyl)-N-(...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311683((S)-1-(3-(2-(2-aminopropanamido)ethyl)phenyl)-N-(2...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311711(CHEMBL1079702 | N-(2-methoxybenzyl)-1-(3-((2-(meth...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311693(CHEMBL1076431 | N-(2-methoxybenzyl)-1-(3-(1-(2-(me...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase SETD7(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311688(CHEMBL1080460 | N-(2-methoxybenzyl)-1-(3-((2-(meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human recombinant SET7/9 expressed in Escherichia coli by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311688(CHEMBL1080460 | N-(2-methoxybenzyl)-1-(3-((2-(meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PRMT1 expressed in Escherichia coli by microbeta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed