Compile Data Set for Download or QSAR
maximum 50k data
Found 56 Enz. Inhib. hit(s) with all data for entry = 3460
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35079(N-acylpolyamine (NAPA) scaffold, 26)
Affinity DataIC50:  2.30E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35078(N-acylpolyamine (NAPA) scaffold, 25)
Affinity DataIC50:  2.60E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35078(N-acylpolyamine (NAPA) scaffold, 25)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35076(N-acylpolyamine (NAPA) scaffold, 23)
Affinity DataIC50:  2.80E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35077(N-acylpolyamine (NAPA) scaffold, 24)
Affinity DataIC50:  2.80E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35080(N-acylpolyamine (NAPA) scaffold, 27)
Affinity DataIC50:  2.90E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35079(N-acylpolyamine (NAPA) scaffold, 26)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35076(N-acylpolyamine (NAPA) scaffold, 23)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35080(N-acylpolyamine (NAPA) scaffold, 27)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35083(N-acylpolyamine (NAPA) scaffold, 34)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35071(N-acylpolyamine (NAPA) scaffold, 18)
Affinity DataIC50:  6.40E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35071(N-acylpolyamine (NAPA) scaffold, 18)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35074(N-acylpolyamine (NAPA) scaffold, 21)
Affinity DataIC50:  6.60E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35077(N-acylpolyamine (NAPA) scaffold, 24)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35070(N-acylpolyamine (NAPA) scaffold, 17)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35072(N-acylpolyamine (NAPA) scaffold, 19)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35074(N-acylpolyamine (NAPA) scaffold, 21)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35069(N-acylpolyamine (NAPA) scaffold, 16)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35075(N-acylpolyamine (NAPA) scaffold, 22)
Affinity DataIC50:  8.20E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35070(N-acylpolyamine (NAPA) scaffold, 17)
Affinity DataIC50:  8.20E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35062(N-acylpolyamine (NAPA) scaffold, 9)
Affinity DataIC50:  9.20E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35073(N-acylpolyamine (NAPA) scaffold, 20)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35075(N-acylpolyamine (NAPA) scaffold, 22)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35069(N-acylpolyamine (NAPA) scaffold, 16)
Affinity DataIC50:  1.00E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35072(N-acylpolyamine (NAPA) scaffold, 19)
Affinity DataIC50:  1.05E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35068(N-acylpolyamine (NAPA) scaffold, 15)
Affinity DataIC50:  1.20E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35068(N-acylpolyamine (NAPA) scaffold, 15)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35066(N-acylpolyamine (NAPA) scaffold, 13)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35067(N-acylpolyamine (NAPA) scaffold, 14)
Affinity DataIC50:  1.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35081(N-acylpolyamine (NAPA) scaffold, 28)
Affinity DataIC50:  1.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35066(N-acylpolyamine (NAPA) scaffold, 13)
Affinity DataIC50:  1.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35081(N-acylpolyamine (NAPA) scaffold, 28)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35061(N-acylpolyamine (NAPA) scaffold, 8)
Affinity DataIC50:  1.70E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35073(N-acylpolyamine (NAPA) scaffold, 20)
Affinity DataIC50:  1.70E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35058(N-acylpolyamine (NAPA) scaffold, 5)
Affinity DataIC50:  1.80E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35059(N-acylpolyamine (NAPA) scaffold, 6)
Affinity DataIC50:  2.00E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35067(N-acylpolyamine (NAPA) scaffold, 14)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35062(N-acylpolyamine (NAPA) scaffold, 9)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35063(N-acylpolyamine (NAPA) scaffold, 10)
Affinity DataIC50:  2.40E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35063(N-acylpolyamine (NAPA) scaffold, 10)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35060(N-acylpolyamine (NAPA) scaffold, 7)
Affinity DataIC50:  3.80E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35061(N-acylpolyamine (NAPA) scaffold, 8)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35064(N-acylpolyamine (NAPA) scaffold, 11)
Affinity DataIC50:  4.10E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35083(N-acylpolyamine (NAPA) scaffold, 34)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35057(N-acylpolyamine (NAPA) scaffold, 4)
Affinity DataIC50:  4.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35064(N-acylpolyamine (NAPA) scaffold, 11)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35056(N-acylpolyamine (NAPA) scaffold, 3)
Affinity DataIC50:  6.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35055(N-acylpolyamine (NAPA) scaffold, 2)
Affinity DataIC50:  8.50E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35058(N-acylpolyamine (NAPA) scaffold, 5)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35065(N-acylpolyamine (NAPA) scaffold, 12)
Affinity DataIC50: >1.00E+5nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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