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Found 21 Enz. Inhib. hit(s) with all data for entry = 50030979
LigandPNGBDBM50304703(2-((3R)-1-(aminomethyl)-3-propylcyclopentyl)acetic...)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304707(2-((1R,3R)-1-(aminomethyl)-3-methylcyclopentyl)ace...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304702(2-((3R)-1-(aminomethyl)-3-ethylcyclopentyl)acetic ...)
Affinity DataIC50:  53nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304693(2-(1-(aminomethyl)-3-ethylcyclopentyl)acetic acid ...)
Affinity DataIC50:  55nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304694(2-(1-(aminomethyl)-3-propylcyclopentyl)acetic acid...)
Affinity DataIC50:  69nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304708(2-((1S,3R)-1-(aminomethyl)-3-methylcyclopentyl)ace...)
Affinity DataIC50:  71nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50164279((S)-3-(aminomethyl)-5-methylhexanoic acid | (S)-3-...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304692(2-(1-(aminomethyl)-3-methylcyclopentyl)acetic acid...)
Affinity DataIC50:  82nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304701(2-((3R)-1-(aminomethyl)-3-methylcyclopentyl)acetic...)
Affinity DataIC50:  88nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080153((1-Aminomethyl-cyclohexyl)-acetic acid | 2-(1-(ami...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
LigandPNGBDBM50304691(CHEMBL610734 | Gababutin)
Affinity DataIC50:  420nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304695(2-(1-(aminomethyl)-3-butylcyclopentyl)acetic acid ...)
Affinity DataIC50:  690nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304705(2-((3S)-1-(aminomethyl)-3-ethylcyclopentyl)acetic ...)
Affinity DataIC50:  706nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304696(2-(1-(aminomethyl)-3-isobutylcyclopentyl)acetic ac...)
Affinity DataIC50:  760nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304706(2-((3S)-1-(aminomethyl)-3-propylcyclopentyl)acetic...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304704(2-((3S)-1-(aminomethyl)-3-methylcyclopentyl)acetic...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304690(2-(1-(aminomethyl)-3,3-dimethylcyclopentyl)acetic ...)
Affinity DataIC50:  3.18E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304698(2-(1-(aminomethyl)-3-phenylcyclopentyl)acetic acid...)
Affinity DataIC50:  5.06E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304700(2-(1-(aminomethyl)-3-phenethylcyclopentyl)acetic a...)
Affinity DataIC50:  6.23E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304699(2-(1-(aminomethyl)-3-benzylcyclopentyl)acetic acid...)
Affinity DataIC50:  9.28E+3nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50304697(2-(1-(aminomethyl)-3-tert-butylcyclopentyl)acetic ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]gabapentin from calcium channel alpha2delta in pig cerebral cortex membrane after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed