Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50031378
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312314(3,3'-((6S,24S,26aS,31aS,37S,40S,42aS)-22-(2-amino-...)
Affinity DataKd:  1.06E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312360((S)-5-amino-4-(2-((22aS,27aS,33S,36S,38aS)-7-((S)-...)
Affinity DataKd:  3.20E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312316(3-((6S,9S,11aS,27S,29aS,34aS)-25-(2-amino-2-oxoeth...)
Affinity DataKd:  5.20E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312317(3,3'-((6S,19S,21aS,26aS,32S,35S,37aS,Z)-17-(2-amin...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312318((S)-5-amino-4-(2-((6S,9S,11aS,29aS,34aS)-18-((S)-1...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312319((S)-5-amino-4-(2-((6S,9S,11aS,28aS,33aS)-18-((S)-1...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312320((S)-5-amino-4-(2-((6S,9S,11aS,27aS,32aS)-18-((S)-1...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312321((S)-5-amino-4-(2-((3aS,8aS,22aS,25S,28S)-16-((S)-1...)
Affinity DataKd:  1.71E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312322((S)-5-amino-4-(2-((3aS,8aS,21aS,24S,27S)-15-((S)-1...)
Affinity DataKd:  2.18E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312323(3-((19S,21aS,26aS,32S,35S,37aS)-17-(2-amino-2-oxoe...)
Affinity DataKd:  1.12E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312324(3-((18S,20aS,25aS,31S,34S,36aS)-16-(2-amino-2-oxoe...)
Affinity DataKd:  7.90E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312325(3-((6S,9S,11aS,28S,30aS,35aS)-26-(2-amino-2-oxoeth...)
Affinity DataKd:  1.08E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312326(3-((6S,9S,11aS,26S,28aS,33aS)-24-(2-amino-2-oxoeth...)
Affinity DataKd:  5.70E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312327(3-((6S,9S,11aS,25S,27aS,32aS)-23-(2-amino-2-oxoeth...)
Affinity DataKd:  8.70E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312328((S)-5-amino-4-(2-((6S,20aS,25aS,31S,34S,36aS)-6-(2...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312329(3,3'-((6S,22S,24aS,29aS,35S,38S,40aS,Z)-20-(2-amin...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312330(3,3'-((6S,21S,23aS,28aS,34S,37S,39aS)-19-(2-amino-...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312331(3,3'-((6S,20S,22aS,27aS,33S,36S,38aS)-18-(2-amino-...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312332(3,3'-((6S,18S,20aS,25aS,31S,34S,36aS)-16-(2-amino-...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312333(3,3'-((6S,9S,11aS,17S,28S,30aS,35aS)-26-(2-amino-2...)
Affinity DataKd:  1.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312334((S)-4-(2-((S)-N-allyl-1-((S)-1-((S)-2-((2S,3R)-2-(...)
Affinity DataKd:  5.90E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312335((S)-5-(allyl(2-amino-2-oxoethyl)amino)-4-((S)-1-((...)
Affinity DataKd:  5.30E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312336((S)-5-((S)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-(ally...)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312336((S)-5-((S)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-(ally...)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312337(3,3'-((6S,27S,29aS,34aS,40S,43S,45aS)-25-(2-amino-...)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312338(3,3'-((6S,26S,28aS,33aS,39S,42S,44aS)-24-(2-amino-...)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312339(3,3'-((6S,27S,29aS,34aS,40S,43S,45aS)-25-(2-amino-...)
Affinity DataKd:  1.90E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312340(3,3'-((6S,26S,28aS,33aS,39S,42S,44aS)-24-(2-amino-...)
Affinity DataKd:  2.40E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312341(3,3'-((6S,25S,27aS,32aS,38S,41S,43aS)-23-(2-amino-...)
Affinity DataKd:  3.80E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312342(3-((24S,26aS,31aS,37S,40S,42aS)-22-(2-amino-2-oxoe...)
Affinity DataKd:  3.10E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312343(3-((23S,25aS,30aS,36S,39S,41aS-21-(2-amino-2-oxoet...)
Affinity DataKd:  3.50E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312344((S)-5-amino-4-(2-((3aS,8aS,23aS,26S,29S)-17-((S)-1...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312345(3-((20S,22aS,27aS,33S,36S,38aS)-18-(2-amino-2-oxoe...)
Affinity DataKd:  4.40E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312346(3-((19S,21aS,26aS,32S,35S,37aS)-17-(2-amino-2-oxoe...)
Affinity DataKd:  4.70E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312347(3,3'-((6S,30S,32aS,37aS,43S,46S,48aS)-28-(2-amino-...)
Affinity DataKd:  2.30E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312348(3,3'-((6S,29S,31aS,36aS,42S,45S,47aS)-27-(2-amino-...)
Affinity DataKd:  3.20E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312349(3,3'-((6S,28S,30aS,35aS,41S,44S,46aS)-26-(2-amino-...)
Affinity DataKd:  2.20E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312350(3,3'-((6S,22S,24aS,29aS,35S,38S,40aS)-20-(2-amino-...)
Affinity DataKd:  6.50E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312351((S)-5-amino-4-(2-((6S,21aS,26aS,32S,35S,37aS)-6-(2...)
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312352((S)-5-amino-4-(2-((6S,23aS,28aS,34S,37S,39aS)-6-(2...)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312353((S)-5-amino-4-(2-((6S,24aS,29aS,35S,38S,40aS)-6-(2...)
Affinity DataKd:  3.40E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312354((S)-5-amino-4-(2-((6S,25aS,30aS,36S,39S,41aS)-6-(2...)
Affinity DataKd:  3.50E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312355(3-((21S,23aS,28aS,34S,37S,39aS)-19-(2-amino-2-oxoe...)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312356(3-((22S,24aS,29aS,35S,38S,40aS)-20-(2-amino-2-oxoe...)
Affinity DataKd:  3.40E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312357((S)-5-amino-4-(2-((6S,9S,11aS,29aS,34aS)-18-((S)-1...)
Affinity DataKd:  2.80E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312358((S)-5-amino-4-(2-((20aS,25aS,31S,34S,36aS,Z)-7-((S...)
Affinity DataKd:  3.00E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312359((S)-5-amino-4-(2-((21aS,26aS,32S,35S,37aS)-7-((S)-...)
Affinity DataKd:  3.10E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50312315(CHEMBL1075925 | PEPTAPPEE)
Affinity DataKd:  5.00E+4nMAssay Description:Binding affinity to ubiquitin E2 variant domain of human Tsg101 by fluorescent anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB