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PubMed code 1992129

Compile data set for download or QSAR
Found 27 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM14361
PNG
((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Show SMILES COc1ccc(cc1OC1CCCC1)C1CNC(=O)C1
Show InChI InChI=1S/C16H21NO3/c1-19-14-7-6-11(12-9-16(18)17-10-12)8-15(14)20-13-4-2-3-5-13/h6-8,12-13H,2-5,9-10H2,1H3,(H,17,18)
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n/an/a 2.60n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228824
PNG
(CHEMBL2112408)
Show SMILES COc1ccc(cc1O[C@@H]1CC2CCC1C2)C1CNC(=O)N1C
Show InChI InChI=1S/C18H24N2O3/c1-20-14(10-19-18(20)21)12-5-6-15(22-2)17(9-12)23-16-8-11-3-4-13(16)7-11/h5-6,9,11,13-14,16H,3-4,7-8,10H2,1-2H3,(H,19,21)/t11?,13?,14?,16-/m1/s1
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n/an/a 2.60n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228833
PNG
(CHEMBL318836)
Show SMILES COc1ccc(cc1OC1CC2CC1C=C2)C1CNC(=O)N1C
Show InChI InChI=1S/C18H22N2O3/c1-20-14(10-19-18(20)21)12-5-6-15(22-2)17(9-12)23-16-8-11-3-4-13(16)7-11/h3-6,9,11,13-14,16H,7-8,10H2,1-2H3,(H,19,21)
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n/an/a 3.10n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228829
PNG
(CHEMBL2111611)
Show SMILES COc1ccc(cc1O[C@H]1CC2CCC1C2)C1CNC(=O)N1C
Show InChI InChI=1S/C18H24N2O3/c1-20-14(10-19-18(20)21)12-5-6-15(22-2)17(9-12)23-16-8-11-3-4-13(16)7-11/h5-6,9,11,13-14,16H,3-4,7-8,10H2,1-2H3,(H,19,21)/t11?,13?,14?,16-/m0/s1
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n/an/a 7.70n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228825
PNG
(CHEMBL2112409)
Show SMILES COc1ccc(cc1O[C@@H]1CC2CC1C1CCCC21)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-17(11-22-21(23)24)12-6-7-18(25-2)20(9-12)26-19-10-13-8-16(19)15-5-3-4-14(13)15/h6-7,9,13-17,19H,3-5,8,10-11H2,1-2H3,(H,22,24)/t13?,14?,15?,16?,17?,19-/m1/s1
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n/an/a 10n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228822
PNG
(CHEMBL2112410)
Show SMILES COc1ccc(cc1O[C@@H]1CC2CC1c1ccccc21)C1CNC(=O)N1C
Show InChI InChI=1S/C22H24N2O3/c1-24-18(12-23-22(24)25)13-7-8-19(26-2)21(10-13)27-20-11-14-9-17(20)16-6-4-3-5-15(14)16/h3-8,10,14,17-18,20H,9,11-12H2,1-2H3,(H,23,25)/t14?,17?,18?,20-/m1/s1
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n/an/a 21n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228831
PNG
(CHEMBL2111610)
Show SMILES COc1ccc(cc1O[C@H]1CC2CC1C1CCCC21)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-17(11-22-21(23)24)12-6-7-18(25-2)20(9-12)26-19-10-13-8-16(19)15-5-3-4-14(13)15/h6-7,9,13-17,19H,3-5,8,10-11H2,1-2H3,(H,22,24)/t13?,14?,15?,16?,17?,19-/m0/s1
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n/an/a 23n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228834
PNG
(CHEMBL101172)
Show SMILES COc1ccc(cc1OC1CC2CCC1CC2)C1CNC(=O)N1C
Show InChI InChI=1S/C19H26N2O3/c1-21-15(11-20-19(21)22)14-7-8-16(23-2)18(10-14)24-17-9-12-3-5-13(17)6-4-12/h7-8,10,12-13,15,17H,3-6,9,11H2,1-2H3,(H,20,22)
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n/an/a 81n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228823
PNG
(CHEMBL101504)
Show SMILES COc1ccc(cc1OC1CC2C3CCC(C3)C2C1)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-18(11-22-21(23)24)14-5-6-19(25-2)20(8-14)26-15-9-16-12-3-4-13(7-12)17(16)10-15/h5-6,8,12-13,15-18H,3-4,7,9-11H2,1-2H3,(H,22,24)
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n/an/a>100n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228826
PNG
(CHEMBL317379)
Show SMILES COc1ccc(cc1OC1C2CC3CC(C2)CC1C3)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-17(11-22-21(23)24)14-3-4-18(25-2)19(10-14)26-20-15-6-12-5-13(8-15)9-16(20)7-12/h3-4,10,12-13,15-17,20H,5-9,11H2,1-2H3,(H,22,24)
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n/an/a>100n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228832
PNG
(CHEMBL100679)
Show SMILES COc1ccc(cc1OC1CC2C1C1CCC2C1)C1CNC(=O)N1C
Show InChI InChI=1S/C20H26N2O3/c1-22-15(10-21-20(22)23)12-5-6-16(24-2)17(8-12)25-18-9-14-11-3-4-13(7-11)19(14)18/h5-6,8,11,13-15,18-19H,3-4,7,9-10H2,1-2H3,(H,21,23)
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n/an/a 100n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228830
PNG
(CHEMBL101505)
Show SMILES COc1ccc(cc1OC1CC2CCC(C2)C1)C1CNC(=O)N1C
Show InChI InChI=1S/C19H26N2O3/c1-21-16(11-20-19(21)22)14-5-6-17(23-2)18(10-14)24-15-8-12-3-4-13(7-12)9-15/h5-6,10,12-13,15-16H,3-4,7-9,11H2,1-2H3,(H,20,22)
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n/an/a>100n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to rat cerebral cortex membranes


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228827
PNG
(CHEMBL2111609)
Show SMILES COc1ccc(cc1O[C@H]1CC2CC1c1ccccc21)C1CNC(=O)N1C
Show InChI InChI=1S/C22H24N2O3/c1-24-18(12-23-22(24)25)13-7-8-19(26-2)21(10-13)27-20-11-14-9-17(20)16-6-4-3-5-15(14)16/h3-8,10,14,17-18,20H,9,11-12H2,1-2H3,(H,23,25)/t14?,17?,18?,20-/m0/s1
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Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228833
PNG
(CHEMBL318836)
Show SMILES COc1ccc(cc1OC1CC2CC1C=C2)C1CNC(=O)N1C
Show InChI InChI=1S/C18H22N2O3/c1-20-14(10-19-18(20)21)12-5-6-15(22-2)17(9-12)23-16-8-11-3-4-13(16)7-11/h3-6,9,11,13-14,16H,7-8,10H2,1-2H3,(H,19,21)
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n/an/a 130n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228824
PNG
(CHEMBL2112408)
Show SMILES COc1ccc(cc1O[C@@H]1CC2CCC1C2)C1CNC(=O)N1C
Show InChI InChI=1S/C18H24N2O3/c1-20-14(10-19-18(20)21)12-5-6-15(22-2)17(9-12)23-16-8-11-3-4-13(16)7-11/h5-6,9,11,13-14,16H,3-4,7-8,10H2,1-2H3,(H,19,21)/t11?,13?,14?,16-/m1/s1
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n/an/a 220n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228822
PNG
(CHEMBL2112410)
Show SMILES COc1ccc(cc1O[C@@H]1CC2CC1c1ccccc21)C1CNC(=O)N1C
Show InChI InChI=1S/C22H24N2O3/c1-24-18(12-23-22(24)25)13-7-8-19(26-2)21(10-13)27-20-11-14-9-17(20)16-6-4-3-5-15(14)16/h3-8,10,14,17-18,20H,9,11-12H2,1-2H3,(H,23,25)/t14?,17?,18?,20-/m1/s1
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n/an/a 290n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228829
PNG
(CHEMBL2111611)
Show SMILES COc1ccc(cc1O[C@H]1CC2CCC1C2)C1CNC(=O)N1C
Show InChI InChI=1S/C18H24N2O3/c1-20-14(10-19-18(20)21)12-5-6-15(22-2)17(9-12)23-16-8-11-3-4-13(16)7-11/h5-6,9,11,13-14,16H,3-4,7-8,10H2,1-2H3,(H,19,21)/t11?,13?,14?,16-/m0/s1
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n/an/a 460n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE).


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM14361
PNG
((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Show SMILES COc1ccc(cc1OC1CCCC1)C1CNC(=O)C1
Show InChI InChI=1S/C16H21NO3/c1-19-14-7-6-11(12-9-16(18)17-10-12)8-15(14)20-13-4-2-3-5-13/h6-8,12-13H,2-5,9-10H2,1H3,(H,17,18)
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n/an/a 490n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE)


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228825
PNG
(CHEMBL2112409)
Show SMILES COc1ccc(cc1O[C@@H]1CC2CC1C1CCCC21)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-17(11-22-21(23)24)12-6-7-18(25-2)20(9-12)26-19-10-13-8-16(19)15-5-3-4-14(13)15/h6-7,9,13-17,19H,3-5,8,10-11H2,1-2H3,(H,22,24)/t13?,14?,15?,16?,17?,19-/m1/s1
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n/an/a 490n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228831
PNG
(CHEMBL2111610)
Show SMILES COc1ccc(cc1O[C@H]1CC2CC1C1CCCC21)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-17(11-22-21(23)24)12-6-7-18(25-2)20(9-12)26-19-10-13-8-16(19)15-5-3-4-14(13)15/h6-7,9,13-17,19H,3-5,8,10-11H2,1-2H3,(H,22,24)/t13?,14?,15?,16?,17?,19-/m0/s1
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n/an/a 560n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE).


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228823
PNG
(CHEMBL101504)
Show SMILES COc1ccc(cc1OC1CC2C3CCC(C3)C2C1)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-18(11-22-21(23)24)14-5-6-19(25-2)20(8-14)26-15-9-16-12-3-4-13(7-12)17(16)10-15/h5-6,8,12-13,15-18H,3-4,7,9-11H2,1-2H3,(H,22,24)
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n/an/a 1.40E+3n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228830
PNG
(CHEMBL101505)
Show SMILES COc1ccc(cc1OC1CC2CCC(C2)C1)C1CNC(=O)N1C
Show InChI InChI=1S/C19H26N2O3/c1-21-16(11-20-19(21)22)14-5-6-17(23-2)18(10-14)24-15-8-12-3-4-13(7-12)9-15/h5-6,10,12-13,15-16H,3-4,7-9,11H2,1-2H3,(H,20,22)
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n/an/a 2.40E+3n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228834
PNG
(CHEMBL101172)
Show SMILES COc1ccc(cc1OC1CC2CCC1CC2)C1CNC(=O)N1C
Show InChI InChI=1S/C19H26N2O3/c1-21-15(11-20-19(21)22)14-7-8-16(23-2)18(10-14)24-17-9-12-3-5-13(17)6-4-12/h7-8,10,12-13,15,17H,3-6,9,11H2,1-2H3,(H,20,22)
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n/an/a 2.50E+3n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228832
PNG
(CHEMBL100679)
Show SMILES COc1ccc(cc1OC1CC2C1C1CCC2C1)C1CNC(=O)N1C
Show InChI InChI=1S/C20H26N2O3/c1-22-15(10-21-20(22)23)12-5-6-16(24-2)17(8-12)25-18-9-14-11-3-4-13(7-11)19(14)18/h5-6,8,11,13-15,18-19H,3-4,7,9-10H2,1-2H3,(H,21,23)
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n/an/a 3.10E+3n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50010981
PNG
((Ro 20-1724)4-(3-Butoxy-4-methoxy-benzyl)-imidazol...)
Show SMILES CCCCOc1cc(CC2CNC(=O)N2)ccc1OC
Show InChI InChI=1S/C15H22N2O3/c1-3-4-7-20-14-9-11(5-6-13(14)19-2)8-12-10-16-15(18)17-12/h5-6,9,12H,3-4,7-8,10H2,1-2H3,(H2,16,17,18)
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n/an/a 6.00E+3n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE)


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228827
PNG
(CHEMBL2111609)
Show SMILES COc1ccc(cc1O[C@H]1CC2CC1c1ccccc21)C1CNC(=O)N1C
Show InChI InChI=1S/C22H24N2O3/c1-24-18(12-23-22(24)25)13-7-8-19(26-2)21(10-13)27-20-11-14-9-17(20)16-6-4-3-5-15(14)16/h3-8,10,14,17-18,20H,9,11-12H2,1-2H3,(H,23,25)/t14?,17?,18?,20-/m0/s1
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n/an/a 1.00E+4n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE).


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4C


(Rattus norvegicus)
BDBM50228826
PNG
(CHEMBL317379)
Show SMILES COc1ccc(cc1OC1C2CC3CC(C2)CC1C3)C1CNC(=O)N1C
Show InChI InChI=1S/C21H28N2O3/c1-23-17(11-22-21(23)24)14-3-4-18(25-2)19(10-14)26-20-15-6-12-5-13(8-15)9-16(20)7-12/h3-4,10,12-13,15-17,20H,5-9,11H2,1-2H3,(H,22,24)
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n/an/a 1.10E+4n/an/an/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Inhibition of calcium-independent Phosphodiesterase 4


J Med Chem 34: 291-8 (1991)


Article DOI: 10.1021/jm00105a045
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%