Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50039032
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305278(CHEMBL595069 | iodoresiniferatoxin)
Affinity DataIC50:  4.00E+3nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305279(CHEMBL595046 | [(1R,2R,6R,10S,11R,13S,15R,17R)-13-...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305280(CHEMBL594862 | [(1R,2R,6R,10S,11R,13S,15R,17R)-13-...)
Affinity DataEC50:  17.4nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305284(CHEMBL593623 | [(1R,2R,6R,10S,11R,13S,15R,17R)-13-...)
Affinity DataEC50:  13.7nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305282(CHEMBL594895 | [(1R,2R,6R,10S,11R,13S,15R,17R)-13-...)
Affinity DataEC50:  0.980nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305285(CHEMBL595262 | [(1R,2R,6R,10S,11R,13S,15R,17R)-13-...)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305283(CHEMBL594016 | [(1R,2R,6R,10S,11R,13S,15R,17R)-13-...)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataEC50:  0.0190nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50305281(CHEMBL594649 | [(1R,2R,6R,10S,11R,13S,15R,17R)-13-...)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed