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Found 15 Enz. Inhib. hit(s) with all data for entry = 50031661
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316843(2-Phenyl-4-(prop-2-yn-1-yloxy)-5,6,7,8-tetrahydro[...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316849(2-(4-Fluorobenzyl)-5,6-dimethyl-3-prop-2-yn-1-ylth...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316851(2-Phenyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316847(2,5,6-Trimethyl-3-prop-2-yn-1-ylthieno[2,3-d]pyrim...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316850(2-Methyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316845(2-Methyl-3-prop-2-yn-1-yl-5, 6, 7, 8-tetrahydro [1...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316846(2-(4-Fluorobenzyl)-3-prop-2-yn-1-yl-5,6,7,8-tetrah...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316850(2-Methyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316846(2-(4-Fluorobenzyl)-3-prop-2-yn-1-yl-5,6,7,8-tetrah...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316848(5,6-Dimethyl-2-phenyl-3-prop-2-yn-1-ylthieno[2, 3-...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316847(2,5,6-Trimethyl-3-prop-2-yn-1-ylthieno[2,3-d]pyrim...)
Affinity DataKi:  3.79E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316849(2-(4-Fluorobenzyl)-5,6-dimethyl-3-prop-2-yn-1-ylth...)
Affinity DataKi:  7.62E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316851(2-Phenyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  9.70E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed