Compile Data Set for Download or QSAR
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Found 35 Enz. Inhib. hit(s) with all data for entry = 50041782
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415454(CHEMBL597559)
Affinity DataKi:  26.9nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415455(CHEMBL603878)
Affinity DataKi:  35.5nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415452(CHEMBL598819)
Affinity DataKi:  93.3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415447(CHEMBL597973)
Affinity DataKi:  93.3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415447(CHEMBL597973)
Affinity DataKi:  93.3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415455(CHEMBL603878)
Affinity DataKi:  95.5nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415454(CHEMBL597559)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415452(CHEMBL598819)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415453(CHEMBL597560)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415455(CHEMBL603878)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415451(CHEMBL597167)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415453(CHEMBL597560)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415458(CHEMBL597955)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415450(CHEMBL597169)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415453(CHEMBL597560)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415452(CHEMBL598819)
Affinity DataKi:  191nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415448(CHEMBL599817)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415460(CHEMBL597580)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415454(CHEMBL597559)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415451(CHEMBL597167)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415448(CHEMBL599817)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415456(CHEMBL597355)
Affinity DataKi:  282nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415457(CHEMBL597354)
Affinity DataKi:  372nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415457(CHEMBL597354)
Affinity DataKi:  389nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415450(CHEMBL597169)
Affinity DataKi:  407nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415459(CHEMBL592653)
Affinity DataKi:  407nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415450(CHEMBL597169)
Affinity DataKi:  479nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415448(CHEMBL599817)
Affinity DataKi:  589nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415449(CHEMBL598584)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415458(CHEMBL597955)
Affinity DataKi:  676nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415457(CHEMBL597354)
Affinity DataKi:  759nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415458(CHEMBL597955)
Affinity DataKi:  813nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415452(CHEMBL598819)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415456(CHEMBL597355)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Porto

Curated by ChEMBL
LigandPNGBDBM50415458(CHEMBL597955)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells by microplate beta scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed